SCHEMBL14965978

SCHEMBL14965978

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(Nc3ccc(C(F)(F)F)cc3)n1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
TRPV1 Q8NER1 2/20 0.39
JAK2 O60674 5/20 0.39
FLT3 P36888 3/20 0.39
MTOR P42345 2/20 0.38
SMG1 Q96Q15 2/20 0.38
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
CCNA1 P78396 1/20 0.37
CLK1 P49759 1/20 0.37
JAK1 P23458 2/20 0.36
TYK2 P29597 2/20 0.36
SCN9A Q15858 2/20 0.36
KCNH2 Q12809 1/20 0.36
PIM1 P11309 1/20 0.36
CDK4 P11802 1/20 0.36
CCND3 P30281 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965593 0.88 MET (0.39) TRPV1KCNH2MCHR1
SCHEMBL14965841 0.87 OGA (0.46)
SCHEMBL14965834 0.78 OGA (0.49)
SCHEMBL14965573 0.78 CHRM1 (0.50) KCNH2MCHR1
SCHEMBL14965617 0.77 TRPV1 (0.45) TRPV1KCNH2
SCHEMBL14965871 0.77 ALDH1A1 (0.42)
SCHEMBL14965636 0.76 HRH4 (0.47) CDK2GSK3B
SCHEMBL14965789 0.76 CYP1A2 (0.40) MTOR
SCHEMBL14965943 0.76 GBA1 (0.40) KCNH2
SCHEMBL14966207 0.74 CHRM1 (0.37) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed