SCHEMBL14977138

SCHEMBL14977138

CNC(=O)c1c(-c2ccc(C)cc2)nc2sc(-c3cc(C(=O)NC(C)(C)C)ccc3C)cn12

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 4/20 0.35
THRB P10828 1/20 0.34
CNR1 P21554 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
HDAC1 Q13547 1/20 0.33
RIPK2 O43353 1/20 0.33
S100B P04271 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14977606 0.93 MAPK14 (0.41) MAPK14NPC1RAB9AALDH1A1MAPT
SCHEMBL14977598 0.93 CNR1 (0.42) MAPK14NPC1RAB9ALMNACNR1
SCHEMBL14977625 0.93 RIPK2 (0.36) MAPK14NPC1RAB9ALMNAALDH1A1
SCHEMBL14986303 0.90 ROCK2 (0.37) MAPK14LMNATHRBLCK
SCHEMBL14977604 0.88 MAPK14 (0.36) MAPK14MAPT
SCHEMBL14977618 0.87 LHCGR (0.41) MAPK14NPC1RAB9ALMNATP53
SCHEMBL14977610 0.86 DGAT2 (0.38) MAPK14NPC1RAB9ALMNATHRB
SCHEMBL14977581 0.85 MAPK14 (0.39) MAPK14MAPT
SCHEMBL14977569 0.85 MAPK14 (0.37) MAPK14MAPT
SCHEMBL14976867 0.85 ROCK2 (0.38) MAPK14ALDH1A1RIPK2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO claimed
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed