SCHEMBL1503252

SCHEMBL1503252

CNC(=O)c1cnc(C(N)=O)c(COC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.42
SCN9A Q15858 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
PSMD14 O00487 1/20 0.36
STAMBP O95630 1/20 0.36
COPS5 Q92905 1/20 0.36
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
SYK P43405 2/20 0.35
NNMT P40261 2/20 0.35
PLK1 P53350 2/20 0.35
AOC3 Q16853 1/20 0.35
BAZ2B Q9UIF8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16465850 0.77 BACE1 (0.40) CDK8CDK19SYKNNMTLMNA
SCHEMBL27386166 0.72 ICAM1 (0.38) SIRT2SIRT1SIRT3MKNK1MKNK2
SCHEMBL10093229 0.71 PLAU (0.46) PLK1
SCHEMBL28285907 0.71 NNMT (0.41) HPGDSPSMD14STAMBPCOPS5NNMT
SCHEMBL30478243 0.71 NNMT (0.41) HPGDSPSMD14STAMBPCOPS5NNMT
SCHEMBL3950709 0.69 BAZ2B (0.49) HPGDSMKNK1MKNK2PLK1BAZ2B
SCHEMBL26755208 0.68 PLK1 (0.44) HPGDSSCN9ASCN2ASCN3ASCN10A
SCHEMBL1503082 0.68 HPGDS (0.51) HPGDSMKNK1MKNK2NNMT
SCHEMBL1503085 0.67 NNMT (0.40) HPGDSPSMD14STAMBPCOPS5MKNK1
SCHEMBL1503239 0.67 KDM4E (0.45) MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed