SCHEMBL1503085

SCHEMBL1503085

NC(=O)c1cnc(C(N)=O)c(CO)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NNMT P40261 7/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PSMD14 O00487 1/20 0.37
STAMBP O95630 1/20 0.37
COPS5 Q92905 1/20 0.37
HPGDS O60760 1/20 0.36
CHEK2 O96017 2/20 0.36
MKNK1 Q9BUB5 1/20 0.36
FYN P06241 1/20 0.36
LMNA P02545 1/20 0.35
MAP4K4 O95819 1/20 0.35
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28285907 0.85 NNMT (0.41) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL30478243 0.85 NNMT (0.41) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL840723 0.80 NNMT (0.36) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL30617860 0.75 HPGDS (0.36) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL2397267 0.75 NNMT (0.44) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL2219734 0.73 NNMT (0.46) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL1503082 0.72 HPGDS (0.51) NNMTHPGDSCHEK2MKNK1MAP4K4
Hydrochloric Acid SCHEMBL28641941 0.72 NNMT (0.44) NNMTSMN1; SMN2PSMD14STAMBPCOPS5
SCHEMBL27858247 0.70 CYP19A1 (0.47) CHEK2KDM4E
SCHEMBL7720516 0.68 NNMT (0.41) NNMTSMN1; SMN2PSMD14STAMBPCOPS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP claimed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO claimed
US-11931348-B2 Methods of treating elevated plasma cholesterol Montréal Heart Institute (CA) 2024-03-19 US disclosed
US-20230088095-A1 METHODS OF TREATING ELEVATED PLASMA CHOLESTEROL Montréal Heart Institute (CA) 2023-03-23 US disclosed
US-8742123-B2 HIV integrase inhibitors from pyridoxine TAIMED BIOLOGICS, INC. (TW) 2014-06-03 US disclosed
US-20110178120-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA, INC. (CA) 2011-07-21 US disclosed
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178120-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE PNPO, CCNB1, BLVRB NNMT 483/4885SMN1; SMN2 3503/4885PSMD14 3798/4885
US-11931348-B2 Methods of treating elevated plasma cholesterol CETP, LDLR, APOB NNMT 2444/4885SMN1; SMN2 3911/4885PSMD14 4274/4885
US-20230088095-A1 METHODS OF TREATING ELEVATED PLASMA CHOLESTEROL CETP, LDLR, APOB NNMT 2444/4885SMN1; SMN2 3911/4885PSMD14 4274/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.