SCHEMBL1509195

SCHEMBL1509195

CC1(C)O[C@@H]2[C@H](O1)[C@@H](O)C[C@H]2N

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
ACHE P22303 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15698958 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL14709158 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL28489991 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL12280418 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL2362689 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL15859653 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL1834044 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL14709006 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL1255498 1.00 MGAM (0.33) MGAMCA1CA2GAASI
SCHEMBL12910763 1.00 MGAM (0.33) MGAMCA1CA2GAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 170 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2707363-B1 A PROCESS FOR THE PREPARATION OF BENZYL [(3AS,4R,6S,6AR)-6-HYDROXY-2,2- DIMETHYLTETRAHYDRO-3AH-CYCLOPENTA[D][1,3]DIOXOL]-4-YL]CARBAMATE AND INTERMEDIATES IN THE PROCESS ASTRAZENECA AB (SE) 2015-10-21 EP claimed
US-9079873-B2 Process for the preparation of benzyl [(3aS,4R,6S,6aR)-6-hydroxy-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol]-4-yl]carbamate and intermediates in the process ASTRAZENECA AB (SE) 2015-07-14 US claimed
WO-2012063126-A2 IMPROVED PROCESSES FOR PREPARING PURE (3AR,4S,6R,6AS)-6-AMINO-2,2-DIMETHYLTETRAHDRO-3AH-CYCLOPENTA[D] [1,3]-DIOXOL-4-OL AND ITS KEY STARTING MATERIAL ACTAVIS GROUP PTC EHF (IS) 2012-05-18 WO claimed
US-12318388-B2 Pyrimidine derivatives for prevention and treatment of gram-negative bacterial infection, contamination and fouling Université de Liège (BE) 2025-06-03 US disclosed
CN-113329753-B Pyrimidine derivatives for the prevention and treatment of gram-negative bacterial infections, pollution and fouling 列日大学 2024-08-13 CN disclosed
EP-3955929-B1 NEW PYRIMIDINE DERIVATIVES FOR PREVENTION AND TREATMENT OF GRAM-NEGATIVE BACTERIAL INFECTION, CONTAMINATION AND FOULING UNIV LIEGE (BE) 2024-05-15 EP disclosed
CN-111386271-B Pyrimidine derivatives for the prevention and treatment of bacterial infections 列日大学 2023-05-30 CN disclosed
US-20230062975-A1 HEPATITIS B CAPSID ASSEMBLY MODULATORS SPRING MILL PHARMA, INC. 2023-03-02 US disclosed
CN-109890797-B Substituted carbon nucleoside derivatives useful as anticancer agents 辉瑞公司 2023-02-28 CN disclosed
US-11566001-B2 Hepatitis B capsid assembly modulators VenatoRx Pharmaceuticals, Inc. (US) 2023-01-31 US disclosed
EP-3752506-B1 PYRIMIDINE DERIVATIVES FOR PREVENTION AND TREATMENT OF BACTERIAL INFECTIONS UNIV LIEGE (BE) 2022-12-14 EP disclosed
WO-2009064249-A1 A PROCESS FOR THE PREPARATION OF (3AR,4S, 6R, 6AS)-6-AMINO-2, 2- DIMETHYLTETRAHYDRO-3AH-CYCLOPENTA[D] [1,3] DIOXOL-4-OL DIBENZOYL-L-TARTRATE AND TO PRODUCTS OF SAID PROCESS ASTRAZENECA AB (SE) 2009-05-22 WO disclosed
US-20070293513-A1 Cristalline and amorphous form of a triazolo (4,5-d) pyridimine compound ASTRAZENECA AB (SE) 2007-12-20 US disclosed
US-7265124-B2 Cristalline and amorphous form of a triazolo (4,5-D) pyridimine compound ASTRAZENECA AB (SE) 2007-09-04 US disclosed
US-20070173518-A1 CRISTALLINE AND AMORPHOUS FORM OF A TRIAZOLO (4,5-D) PYRIDIMINE COMPOUND ASTRAZENECA AB (SE) 2007-07-26 US disclosed
EP-1289992-B1 NEW CRYSTALLINE FORM OF A TRIAZOLO(4,5-D)PYRIMIDINE COMPOUND ASTRAZENECA AB (SE) 2006-03-15 EP disclosed
US-6974868-B2 Compounds ASTRAZENECA AB (SE) 2005-12-13 US disclosed
EP-1493745-A1 New crystalline and amorphous form of a triazolo(4,5-D)pyrimidine compound AstraZeneca AB (SE) 2005-01-05 EP disclosed
US-20030181469-A1 Crystalline and amorphous form of a triazolo(4,5-d)pyrimidine compound ASTRA ZENCA AB (SE) 2003-09-25 US disclosed
US-20030144305-A1 Novel compounds ASTRAZENECA AB 2003-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070293513-A1 Cristalline and amorphous form of a triazolo (4,5-d) pyridimine compound PNPO, MT-ND5, CYP3A5 MGAM 3644/4885CA1 2843/4885CA2 2163/4885
US-20230062975-A1 HEPATITIS B CAPSID ASSEMBLY MODULATORS HAVCR2, COPB1, HDLBP MGAM 4436/4885CA1 4284/4885CA2 4777/4885
US-11566001-B2 Hepatitis B capsid assembly modulators HAVCR2, COPB1, HDLBP MGAM 4436/4885CA1 4284/4885CA2 4777/4885
US-12318388-B2 Pyrimidine derivatives for prevention and treatment of gram-negative bacterial infection, contamination and fouling PIGS, TYMP, TYMS MGAM 629/4885CA1 4266/4885CA2 3816/4885
US-20030181469-A1 Crystalline and amorphous form of a triazolo(4,5-d)pyrimidine compound TYMP, TYMS, DPYD MGAM 3878/4885CA1 2837/4885CA2 1671/4885
US-20030144305-A1 Novel compounds DPYD, TYMP, NUDT15 MGAM 4083/4885CA1 4780/4885CA2 3739/4885
US-20070173518-A1 CRISTALLINE AND AMORPHOUS FORM OF A TRIAZOLO (4,5-D) PYRIDIMINE COMPOUND MT-ND5, PNPO, PDXK MGAM 3783/4885CA1 3113/4885CA2 2521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.