SCHEMBL150967

SCHEMBL150967

Cc1c(N)ccc(Br)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
TSHR P16473 2/20 0.40
PIK3CA P42336 1/20 0.40
ALDH1A1 P00352 5/20 0.36
TDP1 Q9NUW8 2/20 0.36
KDM1A O60341 2/20 0.35
KCNH2 Q12809 2/20 0.35
KDM1B Q8NB78 2/20 0.35
AXL P30530 1/20 0.32
S100B P04271 1/20 0.32
TP53 P04637 1/20 0.32
THRB P10828 1/20 0.32
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAPT P10636 4/20 0.31
HTT P42858 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
POLB P06746 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11932855 0.81 ALDH1A1 (0.36) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL441345 0.77 KDM1A (0.43) ALDH1A1KDM1AKCNH2KDM1BAXL
SCHEMBL580651 0.77 CYP3A4 (0.46) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL29947309 0.75 CYP3A4 (0.43) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL239637 0.75 KDM1A (0.38) ALDH1A1KDM1AKCNH2KDM1BAXL
SCHEMBL29386666 0.75 KDM1A (0.38) ALDH1A1KDM1AKCNH2KDM1BAXL
SCHEMBL6648558 0.75 CYP3A4 (0.43) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL16805981 0.75 CYP3A4 (0.43) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL584965 0.75 KDM1A (0.33) ALDH1A1KDM1AKCNH2KDM1B
SCHEMBL29636024 0.75 KDM1A (0.33) ALDH1A1KDM1AKCNH2KDM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 230 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US disclosed
EP-4665730-A1 HETEROCYCLIC GLP-1 AGONISTS Gasherbrum Bio, Inc. (US) 2025-12-24 EP disclosed
US-20250282746-A1 HALOGEN-SUBSTITUTED ISOINDOLINE COMPOUND AND USE THEREOF Chengdu Fendi Pharmaceutical Co., Ltd. (CN) 2025-09-11 US disclosed
EP-4594324-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2025-08-06 EP disclosed
US-12365682-B2 Process to make GLP1 RA and intermediates therefor ELI LILLY AND COMPANY (US) 2025-07-22 US disclosed
CN-120247804-A Preparation method of 5-bromo-4-fluoro-1-methylindazole 杭州国瑞生物科技有限公司 2025-07-04 CN disclosed
CN-120129683-A Azole derivatives as SHP2 inhibitors IRBM股份公司 2025-06-10 CN disclosed
WO-2025098515-A1 HETEROCYCLIC DERIVATIVES, COMPOSITIONS AND USES THEREOF DANATLAS PHARMACEUTICALS CO., LTD. (CN) 2025-05-15 WO disclosed
US-12291529-B2 Heterocyclic GLP-1 agonists GASHERBRUM BIO, INC. (US) 2025-05-06 US disclosed
WO-2025059577-A1 SUBSTITUTED AMINOPYRIDINE COMPOUNDS FOR USE AS AKT1 INHIBITORS ATAVISTIK BIO, INC. (US) 2025-03-20 WO disclosed
US-8110578-B2 Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway SIGNAL PHARMACEUTICALS, LLC (US) 2012-02-07 US disclosed
WO-2011137219-A1 INHIBITORS OF PHOSPHOINOSITIDE DEPENDENT KINASE 1 (PDK1) SCHERING CORPORATION (US) 2011-11-03 WO disclosed
EP-2358718-A1 MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY Signal Pharmaceuticals, LLC (US) 2011-08-24 EP disclosed
US-20110137028-A1 METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS SIGNAL PHARMACEUTICALS, LLC 2011-06-09 US disclosed
WO-2011053518-A1 METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS SIGNAL PHARMACEUTICALS, LLC (US) 2011-05-05 WO disclosed
US-20100216781-A1 mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY SIGNAL PHARMACEUTICALS, LLC 2010-08-26 US disclosed
WO-2010062571-A1 MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY SIGNAL PHARMACEUTICALS, LLC (US) 2010-06-03 WO disclosed
EP-0411199-B1 Imino [(3-halogenophenyl)amino] acetic acid derivatives and herbicides containing same SDS BIOTECH CORP (JP) 1994-03-30 EP disclosed
US-5006160-A Nonphytotoxic to rice SDS BIOTECH KABUSHIKI KAISHA (JP) 1991-04-09 US disclosed
EP-0411199-A1 Imino [(3-halogenophenyl)amino] acetic acid derivatives and herbicides containing same SDS BIOTECH K.K. (JP) 1991-02-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250282746-A1 HALOGEN-SUBSTITUTED ISOINDOLINE COMPOUND AND USE THEREOF FLI1, CYP3A7, GTF2I CYP3A4 8/4885TSHR 2221/4885PIK3CA 4364/4885
US-12365682-B2 Process to make GLP1 RA and intermediates therefor GLP1R, GIPR, NPY4R CYP3A4 1397/4885TSHR 253/4885PIK3CA 1058/4885
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS PTPN1, PTPN5, PTPN3 CYP3A4 2873/4885TSHR 445/4885PIK3CA 243/4885
US-20100216781-A1 mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY MTOR, RICTOR, RPTOR CYP3A4 1316/4885TSHR 1474/4885PIK3CA 10/4885
US-20110137028-A1 METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS AGER, GPR119, REL CYP3A4 137/4885TSHR 882/4885PIK3CA 2787/4885
US-12291529-B2 Heterocyclic GLP-1 agonists GLP1R, GIPR, IAPP CYP3A4 3522/4885TSHR 118/4885PIK3CA 1561/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.