SCHEMBL15313792

SCHEMBL15313792

O=C(Nc1ccc(Cl)c(Cl)c1)c1cc(CCc2ccccc2)c(O)c(O)c1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 2/20 0.58
PTGS1 P23219 1/20 0.54
TBXAS1 P24557 1/20 0.54
MAPK1 P28482 1/20 0.54
PTGS2 P35354 1/20 0.54
MAPK14 Q16539 1/20 0.54
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
ALDH1A1 P00352 1/20 0.50
ADRB2 P07550 1/20 0.50
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
ALOX15 P16050 1/20 0.47
HTT P42858 1/20 0.47
FPR2 P25090 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15313788 0.81 BCL2 (0.62) BCL2MAPK1ALDH1A1ADRB2KDM4E
SCHEMBL15313790 0.81 BCL2 (0.58) BCL2RAB9AALDH1A1ADRB2KDM4E
SCHEMBL15313786 0.78 BCL2 (0.67) BCL2MAPK1ALDH1A1ADRB2KDM4E
SCHEMBL15313778 0.77 BCL2 (0.56) BCL2ALDH1A1ADRB2KDM4ELMNA
SCHEMBL15314355 0.77 BCL2 (0.56) BCL2PTGS2NPC1RAB9AALDH1A1
SCHEMBL27502192 0.76 ALDH1A1 (0.67) ALDH1A1ADRB2KDM4ELMNASMN1; SMN2
SCHEMBL15313795 0.76 BCL2 (0.57) BCL2MAPK1NPC1RAB9AALDH1A1
SCHEMBL15313783 0.76 BCL2 (0.59) BCL2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL15313847 0.74 BCL2 (1.00) BCL2RAB9AALDH1A1ADRB2KDM4E
SCHEMBL8768715 0.74 PTGS1 (0.68) PTGS1TBXAS1MAPK1PTGS2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed