SCHEMBL15326689

SCHEMBL15326689

O=Cc1ccc(-c2cc3c(c([N+](=O)[O-])c2OCc2ccccc2)CCCC3)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.40
ALDH1A1 P00352 5/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
POLB P06746 2/20 0.38
MAOB P27338 4/20 0.35
TDP1 Q9NUW8 2/20 0.35
TP53 P04637 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
MAOA P21397 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MGMT P16455 1/20 0.33
PTGES O14684 1/20 0.32
HPD P32754 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27971529 0.98 MAPT (0.40) MAPTALDH1A1HPGDMEN1KMT2A
SCHEMBL15326769 0.87 ALDH1A1 (0.41) MAPTALDH1A1HPGDPOLBTDP1
SCHEMBL27971530 0.86 ALDH1A1 (0.41) MAPTALDH1A1HPGDPOLBTDP1
SCHEMBL27971678 0.79 MAOB (0.35) MAPTPOLBMAOBTDP1LMNA
SCHEMBL27940470 0.74 DHODH (0.44) MAPTHPGDPOLBMAOBTDP1
SCHEMBL27921796 0.73 MAOA (0.36) POLBMAOBMAOAMGMTPTGES
SCHEMBL15326750 0.72 MAOB (0.36) MAPTMEN1KMT2APOLBMAOB
SCHEMBL27921772 0.69 HPD (0.33) MAPTMEN1KMT2AMAOBTDP1
SCHEMBL629645 0.68 POLB (0.42) MAPTMEN1KMT2APOLBMAOB
SCHEMBL8044749 0.68 PIN1 (0.44) MAPTMEN1KMT2APOLBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013152683-A1 BICYCLE SUBSTITUTED PYRAZOLONEAZO DERIVATIVES AND PREPARATION METHOD AND USE THEREOF 齐鲁制药有限公司 (CN) 2013-10-17 WO disclosed