Water

Water

SCHEMBL15421412

CC(Cc1ccc(OCC(=O)O)cc1)NCC(O)c1cccc(Cl)c1.O.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB3 known ✓ P13945 14/20 0.96
ADRB2 known ✓ P07550 11/20 0.96
ADRB1 known ✓ P08588 8/20 0.96
ADRA1D known ✓ P25100 1/20 0.96
ADRA1A known ✓ P35348 1/20 0.96
ADRA1B known ✓ P35368 1/20 0.96
CYP2D6 P10635 2/20 0.96
CYP1A2 P05177 1/20 0.96
CYP2C9 P11712 1/20 0.96
CYP2C19 P33261 1/20 0.96
GLA P06280 1/20 0.80
CYP3A4 P08684 1/20 0.79
HIF1A Q16665 1/20 0.79
SLC2A1 P11166 4/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344462 0.99 ADRB3 (0.98) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL304309 0.98 ADRB3 (1.00) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL3692642 0.98 ADRB3 (1.00) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL304308 0.98 ADRB3 (1.00) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL302998 0.98 ADRB3 (1.00) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL302999 0.98 ADRB3 (1.00) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL6539097 0.92 ADRB3 (0.87) ADRB3ADRB2ADRB1CYP2D6ADRA1D
SCHEMBL6539102 0.92 ADRB3 (0.87) ADRB3ADRB2ADRB1CYP2D6ADRA1D
Hydrochloric Acid SCHEMBL6540037 0.91 ADRB3 (0.86) ADRB3ADRB2ADRB1CYP2D6ADRA1D
Hydrochloric Acid SCHEMBL6540028 0.91 ADRB3 (0.86) ADRB3ADRB2ADRB1CYP2D6ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140024677-A1 METHODS FOR INDUCING MITOCHONDRIAL BIOGENESIS MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2014-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140024677-A1 METHODS FOR INDUCING MITOCHONDRIAL BIOGENESIS TFAM, TXNRD2, CPT1B ADRB3 200/4885ADRB2 195/4885ADRB1 179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.