SCHEMBL15515147

SCHEMBL15515147

O=C(O)c1cc(Nc2ccc(F)cc2F)ccc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
KDM4E B2RXH2 2/20 0.53
POLB P06746 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
MAPK14 Q16539 3/20 0.47
MPO P05164 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
SOS1 Q07889 1/20 0.47
CLCN2 P51788 1/20 0.46
MAPK13 O15264 2/20 0.46
MAPK12 P53778 2/20 0.46
MAPK11 Q15759 2/20 0.46
DHODH Q02127 1/20 0.46
GSK3B P49841 1/20 0.45
FABP3 P05413 1/20 0.45
FABP4 P15090 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12483334 0.85 LMNA (0.51) MAPTKDM4ENPC1RAB9AMAPK14
SCHEMBL12482709 0.84 POLB (0.54) MAPTKDM4EPOLBTDP1NPC1
SCHEMBL28741354 0.83 MPO (0.56) MAPTKDM4EPOLBMAPK14MPO
SCHEMBL13285184 0.78 MPO (0.54) MAPTPOLBMAPK14MPOCLCN2
SCHEMBL786240 0.78 ALDH1A1 (0.63) MAPTKDM4EPOLBTDP1NPC1
SCHEMBL12941890 0.76 DHODH (0.50) MAPTNPC1RAB9AMPOALDH1A1
SCHEMBL4863266 0.76 MAP2K1 (0.51) MAPTMAPK14ALDH1A1GAACLCN2
SCHEMBL5753034 0.76 MAPK14 (0.58) MAPTMAPK14ALDH1A1GAASOS1
SCHEMBL27510760 0.75 MAPK13 (0.72) MAPTPOLBNPC1RAB9AMAPK14
SCHEMBL12482895 0.75 P2RX7 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140073651-A1 BENZAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD. (CH) 2014-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140073651-A1 BENZAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS P2RX3, P2RX7, P2RX1 MAPT 4210/4885KDM4E 2905/4885POLB 4438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.