SCHEMBL15524943

SCHEMBL15524943

NS(=O)(=O)c1cc(Br)cnc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.46
KMT2A Q03164 4/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 3/20 0.40
NPC1 O15118 1/20 0.39
POLB P06746 2/20 0.38
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
CA1 P00915 6/20 0.37
CA2 P00918 6/20 0.37
CA4 P22748 4/20 0.37
CA6 P23280 3/20 0.37
CA9 Q16790 3/20 0.37
CA12 O43570 2/20 0.37
CA5A P35218 2/20 0.37
CA7 P43166 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA5B Q9Y2D0 2/20 0.37
CA3 P07451 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789628 0.82 ALPL (0.47) ALPLKMT2AHTTMEN1NPC1
SCHEMBL8515696 0.81 ALPL (0.46) ALPLKMT2AHTTMEN1NPC1
SCHEMBL925314 0.81 ALPL (0.46) ALPLKMT2AHTTMEN1NPC1
Hydrochloric Acid SCHEMBL28094438 0.79 ALPL (0.45) ALPLKMT2AMEN1NPC1POLB
SCHEMBL393051 0.78 KMT2A (0.57) KMT2AHTTMEN1NPC1POLB
SCHEMBL30989718 0.78 ALPL (0.44) ALPLKMT2AMEN1NPC1POLB
SCHEMBL25886719 0.78 ALPL (0.44) ALPLKMT2AMEN1NPC1POLB
SCHEMBL13822303 0.77 NPC1 (0.45) KMT2AHTTMEN1NPC1POLB
SCHEMBL1502723 0.77 KMT2A (0.41) KMT2AHTTMEN1NPC1ALDH1A1
SCHEMBL29469913 0.77 ALDH1A1 (0.48) POLBALDH1A1MAPTCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12187742-B2 Dual ATM and DNA-PK inhibitors for use in anti-tumor therapy XRAD THERAPEUTICS, INC. (US) 2025-01-07 US disclosed
CN-114984003-B Aromatic sulfonamide derivatives 拜耳制药股份公司 2024-08-27 CN disclosed
CN-115054600-B Aromatic sulfonamide derivatives 拜耳制药股份公司 2024-06-14 CN disclosed
CN-112469720-B Dual ATM and DNA-PK inhibitors for use in anti-tumor therapy 艾科思莱德制药公司 2024-03-29 CN disclosed
EP-4327877-A2 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRad Therapeutics, Inc. (US) 2024-02-28 EP disclosed
EP-4327877-A2 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRad Therapeutics, Inc. (US) 2024-02-28 EP disclosed
EP-3784671-B1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRAD THERAPEUTICS INC (US) 2023-10-11 EP disclosed
EP-3784671-B1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRAD THERAPEUTICS INC (US) 2023-10-11 EP disclosed
US-11524938-B2 Aromatic sulfonamide derivatives BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-12-13 US disclosed
US-20220324807-A1 AROMATIC SULFONAMIDE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-10-13 US disclosed
US-20160102051-A1 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS AND VIRAL INFECTIONS ATXA THERAPEUTICS LIMITED (IE) 2016-04-14 US disclosed
US-20160102051-A1 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS AND VIRAL INFECTIONS ATXA THERAPEUTICS LIMITED (IE) 2016-04-14 US disclosed
US-20160016900-A1 THROMBOXANE RECEPTOR ANTAGONISTS ATXA THERAPEUTICS LIMITED (IE) 2016-01-21 US disclosed
US-20160016900-A1 THROMBOXANE RECEPTOR ANTAGONISTS ATXA THERAPEUTICS LIMITED (IE) 2016-01-21 US disclosed
US-20160016900-A1 THROMBOXANE RECEPTOR ANTAGONISTS ATXA THERAPEUTICS LIMITED (IE) 2016-01-21 US disclosed
EP-2838519-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS AND VIRAL INFECTIONS University College Dublin National University Of Ireland, Dublin (IE) 2015-02-25 EP disclosed
EP-2838520-A2 THROMBOXANE RECEPTOR ANTAGONISTS University College Dublin National University Of Ireland, Dublin (IE) 2015-02-25 EP disclosed
WO-2013156871-A9 THROMBOXANE RECEPTOR ANTAGONISTS UNIVERSITY COLLEGE DUBLIN, NATIONAL UNIVERSITY OF IRELAND, DUBLIN (IE) 2015-01-08 WO disclosed
WO-2013156871-A2 THROMBOXANE RECEPTOR ANTAGONISTS UNIVERSITY COLLEGE DUBLIN, NATIONAL UNIVERSITY OF IRELAND, DUBLIN (IE) 2013-10-24 WO disclosed
WO-2013156861-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS AND VIRAL INFECTIONS UNIVERSITY COLLEGE DUBLIN, NATIONAL UNIVERSITY OF IRELAND, DUBLIN (IE) 2013-10-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220324807-A1 AROMATIC SULFONAMIDE DERIVATIVES ARSA, SULT2A1, TPST2 ALPL 2588/4885KMT2A 1375/4885HTT 356/4885
US-20160102051-A1 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS AND VIRAL INFECTIONS TBXA2R, PTGFR, TBXAS1 ALPL 3903/4885KMT2A 1962/4885HTT 1671/4885
US-11524938-B2 Aromatic sulfonamide derivatives ARSA, SULT2A1, TPST2 ALPL 2588/4885KMT2A 1375/4885HTT 356/4885
US-20160016900-A1 THROMBOXANE RECEPTOR ANTAGONISTS TBXA2R, TBXAS1, PTGIR ALPL 4368/4885KMT2A 2845/4885HTT 1866/4885
US-12187742-B2 Dual ATM and DNA-PK inhibitors for use in anti-tumor therapy ATM, CHEK2, CHEK1 ALPL 2100/4885KMT2A 918/4885HTT 2506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.