SCHEMBL1553334

SCHEMBL1553334

COc1cc(O)ccc1[C@H](O)CNC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADRA1A P35348 1/20 0.42
SYK P43405 1/20 0.40
SERPINE1 P05121 1/20 0.40
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
APP P05067 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
DRD2 P14416 2/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1554860 0.85 NQO2 (0.44) NQO2LMNATSHRSYKSERPINE1
SCHEMBL4582959 0.84 DRD2 (0.49) LMNACYP1A2TSHRCYP2C19ADORA3
SCHEMBL1554728 0.81 SYK (0.47) LMNACYP1A2TSHRCYP2C19ADORA3
SCHEMBL1554044 0.80 CA1 (0.47) LMNASYKCTSSCTSK
SCHEMBL1553332 0.78 GPR88 (0.40) NQO2ALDH1A1GAAAPPCTSS
SCHEMBL2011966 0.77 SMN1; SMN2 (0.51) NQO2LMNATSHRSYKSERPINE1
SCHEMBL1553366 0.77 SMN1; SMN2 (0.51) NQO2LMNATSHRSYKSERPINE1
SCHEMBL9149377 0.77 SERPINE1 (0.44) NQO2LMNATSHRSYKSERPINE1
SCHEMBL13997819 0.77 DRD2 (0.42) LMNACYP1A2TSHRCYP2C19ADORA3
SCHEMBL2940084 0.76 NQO2 (0.48) NQO2ALDH1A1GAAAPPDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486030-A1 MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88 Bristol-Myers Squibb Company (US) 2012-08-15 EP disclosed
WO-2011044195-A1 MODULATORS OF G PROTEIN-COUPLED RECEPTOR 88 BRISTOL-MYERS SQUIBB COMPANY (US) 2011-04-14 WO disclosed