SCHEMBL15539246

SCHEMBL15539246

CC(C)(F)CN1CCC(COc2ccc(-c3ccc(C(=O)NC(=O)[C@@H]4CCCN4)cc3)cn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 7/20 0.39
WNT1 P04628 3/20 0.39
LIPE Q05469 1/20 0.38
ACHE P22303 2/20 0.36
HPGDS O60760 1/20 0.36
GSK3B P49841 3/20 0.36
CTSS P25774 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
GPR119 Q8TDV5 1/20 0.35
DPP4 P27487 3/20 0.35
DPP8 Q6V1X1 1/20 0.35
ATM Q13315 1/20 0.35
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15538527 0.98 LIPE (0.39) DYRK1AWNT1LIPEACHEHPGDS
SCHEMBL15539034 0.94 LIPE (0.37) DYRK1AWNT1LIPEACHEHPGDS
SCHEMBL15539677 0.91 DYRK1A (0.37) DYRK1AWNT1LIPEHPGDSGSK3B
SCHEMBL15538470 0.89 SCN9A (0.36) DYRK1AWNT1ACHEHPGDSGSK3B
SCHEMBL15539766 0.89 WDR5 (0.38) DYRK1AWNT1LIPEGSK3B
SCHEMBL15538813 0.89 WDR5 (0.38) DYRK1AWNT1LIPEGSK3B
SCHEMBL15539503 0.89 DYRK1A (0.41) DYRK1AWNT1GSK3BCTSSATM
SCHEMBL15539973 0.88 LIPE (0.37) DYRK1AWNT1LIPEHPGDSGSK3B
SCHEMBL15538893 0.88 LIPE (0.37) DYRK1AWNT1LIPEHPGDSGSK3B
SCHEMBL15539527 0.87 WNT1 (0.38) DYRK1AWNT1LIPEACHEGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2858986-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST Chong Kun Dang Pharmaceutical Corp. (KR) 2015-04-15 EP claimed
WO-2013187646-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2013-12-19 WO claimed
EP-2858986-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST Chong Kun Dang Pharmaceutical Corp. (KR) 2015-04-15 EP disclosed
WO-2013187646-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2013-12-19 WO disclosed