SCHEMBL15544668

SCHEMBL15544668

Cc1ccc2c(c1)NCC2C(=O)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
P2RX7 Q99572 2/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
P2RX5 Q93086 1/20 0.41
P2RX4 Q99571 1/20 0.41
P2RX2 Q9UBL9 1/20 0.41
NPC1 O15118 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
ATM Q13315 1/20 0.38
EPHX2 P34913 1/20 0.38
CYP17A1 P05093 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15544852 0.89 LMNA (0.43) ALDH1A1LMNAP2RX7RAB9ASMN1; SMN2
SCHEMBL15545277 0.82 SMN1; SMN2 (0.47) P2RX7SMN1; SMN2P2RX4MEN1KMT2A
SCHEMBL15545467 0.82 KCNH2 (0.41) ALDH1A1P2RX7RAB9AKDM4EHPGD
SCHEMBL15545879 0.81 ALDH1A1 (0.44) ALDH1A1LMNAP2RX7RAB9ASMN1; SMN2
SCHEMBL15545602 0.80 ALDH1A1 (0.35) ALDH1A1LMNAP2RX7SMN1; SMN2CYP17A1
SCHEMBL15544370 0.77 CNR2 (0.41) ALDH1A1LMNAP2RX7SMN1; SMN2CYP17A1
SCHEMBL15545052 0.77 P2RX4 (0.39) ALDH1A1LMNAP2RX7P2RX5P2RX4
SCHEMBL15545061 0.77 P2RX7 (0.41) ALDH1A1LMNAP2RX7RAB9ASMN1; SMN2
SCHEMBL15545632 0.77 P2RX7 (0.41) ALDH1A1LMNAP2RX7RAB9ASMN1; SMN2
SCHEMBL15544368 0.74 ALDH1A1 (0.44) ALDH1A1LMNAP2RX7SMN1; SMN2P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870139-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
WO-2014005968-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed