SCHEMBL15545602

SCHEMBL15545602

O=C(C1CNc2cc(F)c(F)cc21)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
P2RX7 Q99572 4/20 0.35
LMNA P02545 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
CYP17A1 P05093 1/20 0.33
CYP19A1 P11511 1/20 0.33
POLB P06746 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
CNR2 P34972 1/20 0.32
GRM1 Q13255 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15544370 0.84 CNR2 (0.41) ALDH1A1P2RX7LMNAKCNQ3KCNQ2
SCHEMBL15544852 0.80 LMNA (0.43) ALDH1A1P2RX7LMNASMN1; SMN2NPSR1
SCHEMBL15544668 0.80 ALDH1A1 (0.43) ALDH1A1P2RX7LMNASMN1; SMN2NPSR1
SCHEMBL15545052 0.78 P2RX4 (0.39) ALDH1A1P2RX7LMNACYP17A1CYP19A1
SCHEMBL15544868 0.78 KCNQ3 (0.35) ALDH1A1P2RX7LMNAKCNQ3KCNQ2
SCHEMBL15545277 0.78 SMN1; SMN2 (0.47) P2RX7KCNQ3KCNQ2SMN1; SMN2CYP17A1
SCHEMBL15545467 0.77 KCNH2 (0.41) ALDH1A1P2RX7CYP17A1CYP19A1CNR2
SCHEMBL15545879 0.75 ALDH1A1 (0.44) ALDH1A1P2RX7LMNASMN1; SMN2NPSR1
SCHEMBL15544368 0.75 ALDH1A1 (0.44) ALDH1A1P2RX7LMNASMN1; SMN2NPSR1
SCHEMBL15545182 0.69 KCNH2 (0.42) ALDH1A1LMNACYP17A1CYP19A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870139-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
WO-2014005968-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed