SCHEMBL15545467

SCHEMBL15545467

O=C(C1CNc2ccccc21)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.41
CNR2 P34972 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP17A1 P05093 2/20 0.40
CYP19A1 P11511 2/20 0.40
KDM4E B2RXH2 2/20 0.40
P2RX7 Q99572 2/20 0.39
IDH1 O75874 1/20 0.39
HPGD P15428 1/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.38
XBP1 P17861 1/20 0.38
AGTR1 P30556 1/20 0.37
OPRK1 P41145 1/20 0.37
RECQL P46063 1/20 0.37
RAB9A P51151 1/20 0.37
IDO1 P14902 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545182 0.90 KCNH2 (0.42) KCNH2CNR2ALDH1A1CYP17A1CYP19A1
SCHEMBL15546001 0.87 SMN1; SMN2 (0.46) KCNH2CNR2ALDH1A1KDM4EP2RX7
SCHEMBL15544852 0.82 LMNA (0.43) ALDH1A1CYP17A1CYP19A1KDM4EP2RX7
SCHEMBL15544668 0.82 ALDH1A1 (0.43) ALDH1A1CYP17A1CYP19A1KDM4EP2RX7
SCHEMBL15545052 0.81 P2RX4 (0.39) CNR2ALDH1A1CYP17A1CYP19A1KDM4E
SCHEMBL15544370 0.81 CNR2 (0.41) CNR2ALDH1A1CYP17A1CYP19A1P2RX7
SCHEMBL15544373 0.79 FAAH (0.48) CNR2ALDH1A1KDM4EHPGDMAPT
SCHEMBL15545061 0.78 P2RX7 (0.41) CNR2ALDH1A1P2RX7MAPTRAB9A
SCHEMBL15545632 0.78 P2RX7 (0.41) CNR2ALDH1A1P2RX7IDH1MAPT
SCHEMBL15545277 0.78 SMN1; SMN2 (0.47) CNR2CYP17A1CYP19A1KDM4EP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870139-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
WO-2014005968-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed