SCHEMBL156226

SCHEMBL156226

CCC(CC)(OS(=O)(=O)c1ccc(C)cc1)P(=O)(O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.41
CA12 O43570 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 1/20 0.41
ALDH1A1 P00352 5/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
PTPN1 P18031 1/20 0.39
GAA P10253 3/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
VDR P11473 1/20 0.36
ENPP1 P22413 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9654540 0.83 CA2 (0.39) CA12CA9ALDH1A1KMT2AMEN1
SCHEMBL5324671 0.81 LMNA (0.44) CA12CA9ALDH1A1KMT2AMEN1
SCHEMBL157580 0.80 MMP2 (0.38) MMP2CA12CA9CA14ALDH1A1
SCHEMBL1377737 0.76 MMP2 (0.43) MMP2CA12CA9CA14ALDH1A1
SCHEMBL8394723 0.76 ALDH1A1 (0.44) CA12CA9ALDH1A1KMT2AMEN1
SCHEMBL4195761 0.75 PTPN1 (0.41) ALDH1A1KMT2AMEN1PTPN1GAA
SCHEMBL259737 0.74 MMP2 (0.41) MMP2CA12CA9CA14ALDH1A1
SCHEMBL10572140 0.73 STAT3 (0.44) ALDH1A1KMT2AMEN1GAAENPP1
SCHEMBL2325755 0.73 STAT3 (0.44) ALDH1A1KMT2AMEN1GAAENPP1
SCHEMBL10572152 0.73 STAT3 (0.44) ALDH1A1KMT2AMEN1GAAENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1256585-B1 Process for preparing 9-(2-(diethylphosphonomethoxy)ethyl)-adenine GILEAD SCIENCES INC (US) 2004-09-29 EP claimed
EP-4543859-A1 3-(SULPHONYL OR SULFONIMIDOYL)PROP-2-EN-1-YL]-2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE DERIVATIVES Flindr Therapeutics B.V. (NL) 2025-04-30 EP disclosed
US-20240368204-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF XIZANG HAISCO PHARMACEUTICAL CO., LTD. (CN) 2024-11-07 US disclosed
CN-118488854-A Self-assembling amphiphilic polymers as anti-COVID-19 agents 阿列克斯塞尔公司 2024-08-13 CN disclosed
EP-4353732-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF Xizang Haisco Pharmaceutical Co., Ltd. (CN) 2024-04-17 EP disclosed
WO-2023249490-A1 3-(SULPHONYL OR SULFONIMIDOYL)PROP-2-EN-1-YL]-2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE DERIVATIVES IMMAGENE B.V. (NL) 2023-12-28 WO disclosed
US-11472826-B2 Acyclic antivirals JANSSEN PHARMACEUTICA NV (BE) 2022-10-18 US disclosed
US-20200392169-A1 ACYCLIC ANTIVIRALS JANSSEN BIOPHARMA, LLC 2020-12-17 US disclosed
US-10745427-B2 Acyclic antivirals Janssen Biopharma, Inc. (US) 2020-08-18 US disclosed
US-20190055273-A1 ACYCLIC ANTIVIRALS Janssen Pharmaceuticals, Inc. 2019-02-21 US disclosed
WO-2006130217-A2 SUBSTITUTED PHOSPHATE ESTERS OF NUCLEOSIDE PHOSPHONATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2006-12-07 WO disclosed
US-20050137141-A1 Prodrug composition HILFINGER JOHN (US) 2005-06-23 US disclosed
US-RE38333-E1 Making tenofovir analogs and salts; use as viricides for HIV, retroviruses GILEAD SCIENCES, INC. 2003-11-25 US disclosed
EP-1301519-A2 PRODRUGS OF PHOSPHONATE NUCLEOTIDE ANALOGUES AND METHODS FOR SELECTING AND MAKING SAME GILEAD SCIENCES, INC. (US) 2003-04-16 EP disclosed
WO-2002008241-A2 PRODRUGS OF PHOSPHONATE NUCLEOTIDE ANALOGUES AND METHODS FOR SELECTING AND MAKING SAME GILEAD SCIENCES, INC. (US) 2002-01-31 WO disclosed
US-6069249-A CHEMICAL INTERMEDIATES; DETECTION LABELS FOR NUCLEOTIDE PROBES GILEAD SCIENCES, INC. (US) 2000-05-30 US disclosed
US-5686629-A CHEMICAL INTERMEDIATES GILEAD SCIENCES, INC. (US) 1997-11-11 US disclosed
US-5514798-A REACTION OF CYCLIC CARBONATE WITH PURINE OR PYRIMIDINE BASE IN SOLVENT AND CRYSTALLIZATION GILEAD SCIENCES, INC. (US) 1996-05-07 US disclosed
EP-0550574-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1993-07-14 EP disclosed
WO-1992005180-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11472826-B2 Acyclic antivirals PNP, DUT, TYMP MMP2 3529/4885CA12 4723/4885CA9 4448/4885
US-20240368204-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF ENTPD5, ENTPD1, ENTPD2 MMP2 595/4885CA12 740/4885CA9 349/4885
US-20190055273-A1 ACYCLIC ANTIVIRALS PNP, TYMP, DUT MMP2 3224/4885CA12 4719/4885CA9 4477/4885
US-20200392169-A1 ACYCLIC ANTIVIRALS PNP, DUT, TYMP MMP2 3529/4885CA12 4723/4885CA9 4448/4885
US-20050137141-A1 Prodrug composition CYP3A5, SLC35B2, SLC1A5 MMP2 451/4885CA12 2806/4885CA9 1108/4885
US-10745427-B2 Acyclic antivirals PNP, DUT, TYMP MMP2 3529/4885CA12 4723/4885CA9 4448/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.