Eprosartan

Eprosartan

SCHEMBL156290

CCCCc1ncc(/C=C(/Cc2cccs2)C(=O)O)n1Cc1ccc(C(=O)O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

AGTR1

The experimentally established mechanism targets of Eprosartan. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 known ✓ P30556 2/20 1.00
ABCC3 O15438 1/20 1.00
ABCC2 Q92887 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eprosartan SCHEMBL1815060 1.00 AGTR1 (1.00) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL4026 1.00 AGTR1 (1.00) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL4025 1.00 AGTR1 (1.00) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL7405237 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL1119964 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL1119965 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL7405236 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL1897811 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL6747994 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2
Eprosartan SCHEMBL6747993 0.99 AGTR1 (0.98) AGTR1ABCC3ABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200276166-A1 METHODS OF TREATING NEUROLOGICAL DISORDERS UNIV CALIFORNIA (US) 2020-09-03 US claimed
US-20160367530-A1 METHODS OF TREATING NEUROLOGICAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2016-12-22 US claimed
US-20130066252-A1 METHOD FOR DIAGNOSIS FOR MULTIPLE SCLEROSIS INVOLVING ANTI1-RECEPTOR ANTIBODY CELLTREND GMBH (DE) 2013-03-14 US claimed
US-20120058949-A1 Methods of Treating Neurological Disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2012-03-08 US claimed
US-20100098688-A1 METHOD FOR DIAGNOSIS OF A DISEASE INVOLVING AN ANTI-AT1-RECEPTOR ANTIBODY CELLTREND GMBH (DE) 2010-04-22 US claimed
EP-1884775-A1 Method for diagnosis of a disease involving an anti-AT1-receptor antibody Celltrend GmbH (DE) 2008-02-06 EP claimed
US-20200276166-A1 METHODS OF TREATING NEUROLOGICAL DISORDERS UNIV CALIFORNIA (US) 2020-09-03 US disclosed
US-10668049-B2 Methods of treating cognitive decline with transforming growth factor beta inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-06-02 US disclosed
US-20160367530-A1 METHODS OF TREATING NEUROLOGICAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2016-12-22 US disclosed
US-9468649-B2 Methods of treating epilepsy with transforming growth factor beta inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-18 US disclosed
EP-2558856-B1 METHOD FOR DIAGNOSIS OF MULTIPLE SCLEROSIS INVOLVING ANTI-AT1-RECEPTOR ANTIBODY CELLTREND GMBH (DE) 2016-04-06 EP disclosed
US-20160081901-A1 COMPOSITIONS AND METHODS FOR HAIR GROWTH WUHAN OPTICS VALLEY BRIDGEBIOMED INTERNATIONAL CORPORATION (CN) 2016-03-24 US disclosed
US-20150119329-A1 MODULATION OF ANGIOTENSIN II RECEPTORS FOR THE PREVENTION AND TREATMENT OF MALARIA CEREBRAL NEW YORK UNIVERSITY (US) 2015-04-30 US disclosed
US-20100331356-A1 SELF-MICROEMULSIFYING DRUG DELIVERY SYSTEMS LEK PHARMACEUTICALS D.D. (SI) 2010-12-30 US disclosed
US-7858611-B2 Neurogenesis by modulating angiotensin BRAINCELLS INC. (US) 2010-12-28 US disclosed
US-20100098688-A1 METHOD FOR DIAGNOSIS OF A DISEASE INVOLVING AN ANTI-AT1-RECEPTOR ANTIBODY CELLTREND GMBH (DE) 2010-04-22 US disclosed
EP-2021000-A2 NEUROGENESIS BY MODULATING ANGIOTENSIN Braincells, Inc. (US) 2009-02-11 EP disclosed
US-20080167291-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN BRAINCELLS, INC. (US) 2008-07-10 US disclosed
EP-1884775-A1 Method for diagnosis of a disease involving an anti-AT1-receptor antibody Celltrend GmbH (DE) 2008-02-06 EP disclosed
WO-2007134136-A2 NEUROGENESIS BY MODULATING ANGIOTENSIN BRAINCELLS, INC. (US) 2007-11-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160081901-A1 COMPOSITIONS AND METHODS FOR HAIR GROWTH AGTR2, AGTR1, BDKRB2 AGTR1 2/4885ABCC3 3693/4885ABCC2 3119/4885
US-20150119329-A1 MODULATION OF ANGIOTENSIN II RECEPTORS FOR THE PREVENTION AND TREATMENT OF MALARIA CEREBRAL AGTR2, AGTR1, ACE2 AGTR1 2/4885ABCC3 845/4885ABCC2 494/4885
US-20080167291-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN DCX, NGF, BDNF AGTR1 8/4885ABCC3 4434/4885ABCC2 4558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.