Amphetamine

Amphetamine

SCHEMBL157108

CC(N)Cc1ccccc1.NC(=O)O

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC6A2SLC6A3

The experimentally established mechanism targets of Amphetamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 3/20 0.79
SLC6A3 known ✓ Q01959 1/20 0.79
TAAR1 Q96RJ0 5/20 0.79
SLC6A4 P31645 3/20 0.79
MAOA P21397 1/20 0.79
SIGMAR1 Q99720 1/20 0.79
CYP2A6 P11509 1/20 0.79
ADORA2A P29274 1/20 0.79
ADORA1 P30542 1/20 0.79
ALPI P09923 1/20 0.59
PKM P14618 1/20 0.59
PTGS1 P23219 1/20 0.59
XIAP P98170 1/20 0.59
SLC7A5 Q01650 1/20 0.59
CYP2D6 P10635 1/20 0.55
EPHX1 P07099 2/20 0.53
SLC1A3 P43003 1/20 0.53
SLC1A2 P43004 1/20 0.53
SLC1A1 P43005 1/20 0.53
NPC1 O15118 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amphetamine SCHEMBL29102142 1.00 TAAR1 (0.79) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL29102157 0.92 TAAR1 (0.79) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL27293366 0.92 TAAR1 (0.79) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL8589685 0.92 TAAR1 (0.79) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL3513103 0.90 TAAR1 (0.70) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL29127738 0.90 TAAR1 (0.76) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL28990193 0.89 TAAR1 (0.91) TAAR1SLC6A2SLC6A4MAOASLC6A3
Levamfetamine SCHEMBL9673275 0.89 SLC6A2 (1.00) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL13747801 0.89 SLC6A2 (1.00) TAAR1SLC6A2SLC6A4MAOASLC6A3
Amphetamine SCHEMBL1560962 0.89 SLC6A2 (1.00) TAAR1SLC6A2SLC6A4MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250320178-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2025-10-16 US claimed
US-12427122-B2 Method of making transdermal amphetamine composition with low levels of carbamate NOVEN PHARMACEUTICALS, INC. (US) 2025-09-30 US claimed
US-20240327337-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2024-10-03 US claimed
CN-117529665-A Amphetamine carbamate compounds and methods 诺芬药品公司 2024-02-06 CN claimed
EP-4274555-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2023-11-15 EP claimed
EP-4275055-A2 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2023-11-15 EP claimed
CN-116997330-A Transdermal amphetamine compositions with low levels of carbamate 诺芬药品公司 2023-11-03 CN claimed
US-20230201139-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2023-06-29 US claimed
US-11572339-B2 Amphetamine carbamate compounds and methods NOVEN PHARMACEUTICALS, INC. (US) 2023-02-07 US claimed
US-20220218628-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2022-07-14 US claimed
WO-2022150430-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2022-07-14 WO claimed
WO-2022150431-A2 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2022-07-14 WO claimed
US-20220213029-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2022-07-07 US claimed
US-20260102362-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2026-04-16 US disclosed
US-20260102362-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE NOVEN PHARMACEUTICALS, INC. (US) 2026-04-16 US disclosed
US-20250320178-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS NOVEN PHARMACEUTICALS, INC. (US) 2025-10-16 US disclosed
WO-2012031125-A2 REVERSAL OF GENERAL ANESTHESIA BY ADMINISTRATION OF METHYLPHENIDATE, AMPHETAMINE, MODAFINIL, AMANTADINE, AND/OR CAFFEINE THE GENERAL HOSPITAL CORPORATION (US) 2012-03-08 WO disclosed
US-20110021564-A1 METHOD OF TREATING BINGE EATING DISORDER AND OBESITY RESULTING FROM BINGE EATING BEHAVIOR LCS GROUP, LLC (US) 2011-01-27 US disclosed
US-20100166889-A1 METHOD OF TREATING DEPRESSIVE DISORDERS LCS GROUP, LLC (US) 2010-07-01 US disclosed
WO-2009035473-A2 METHOD OF TREATING BINGE EATING DISORDER, OBESITY RESULTING FROM BINGE EATING BEHAVIOR AND DEPRESSIVE DISORDERS SANFILIPPO LOUIS C (US) 2009-03-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240327337-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS CHAT, CES2, NAAA SLC6A2 98/4885SLC6A3 14/4885TAAR1 97/4885
US-20260102362-A1 TRANSDERMAL AMPHETAMINE COMPOSITIONS WITH LOW LEVELS OF CARBAMATE SLC6A2, SLC6A3, CHAT SLC6A2 1/4885SLC6A3 2/4885TAAR1 72/4885
US-20220213029-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS CHAT, CES2, NAAA SLC6A2 98/4885SLC6A3 14/4885TAAR1 97/4885
US-20110021564-A1 METHOD OF TREATING BINGE EATING DISORDER AND OBESITY RESULTING FROM BINGE EATING BEHAVIOR COMT, MC4R, SLC6A4 SLC6A2 38/4885SLC6A3 6/4885TAAR1 229/4885
US-20100166889-A1 METHOD OF TREATING DEPRESSIVE DISORDERS HTR5A, SLC6A4, HTR4 SLC6A2 7/4885SLC6A3 12/4885TAAR1 107/4885
US-11572339-B2 Amphetamine carbamate compounds and methods CHAT, CES2, NAAA SLC6A2 98/4885SLC6A3 14/4885TAAR1 97/4885
US-20250320178-A1 AMPHETAMINE CARBAMATE COMPOUNDS AND METHODS CHAT, CES2, NAAA SLC6A2 98/4885SLC6A3 14/4885TAAR1 97/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.