SCHEMBL15748380

SCHEMBL15748380

CC(=O)NC1COC/C=C\COCC(C(N)=O)NC(=O)C(CC(N)=O)NC(=O)C(CC(=O)O)NC(=O)C(Cc2ccc(O)cc2)NC(=O)CNC(=O)C(CCC(=O)O)NC(=O)C(Cc2ccccc2)NC1=O

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRB7 Q14451 2/20 0.70
ITGB3 P05106 5/20 0.49
ITGA2B P08514 5/20 0.49
KEAP1 Q14145 1/20 0.47
OPRM1 P35372 2/20 0.46
OPRD1 P41143 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15748405 0.76 GRB7 (0.85) GRB7ITGB3ITGA2BKEAP1
SCHEMBL15748376 0.73 GRB7 (0.72) GRB7ITGB3ITGA2B
SCHEMBL31060478 0.73 ITGB3 (0.56) GRB7ITGB3ITGA2B
SCHEMBL22872704 0.69 ITGB3 (0.59) ITGB3ITGA2B
SCHEMBL22342240 0.69 KEAP1 (0.63) KEAP1
SCHEMBL13573536 0.68 ITGB3 (0.51) GRB7ITGB3ITGA2B
SCHEMBL22342263 0.68 KEAP1 (0.63) ITGB3ITGA2BKEAP1
SCHEMBL16576430 0.68 OXTR (0.51) GRB7ITGB3ITGA2B
SCHEMBL16135323 0.68 ITGB3 (0.54) ITGB3ITGA2B
SCHEMBL30389411 0.68 FLT1 (0.49) GRB7OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014078889-A1 IMPROVED INHIBITORS OF GRB7 MONASH UNIVERSITY (AU) 2014-05-30 WO disclosed