Bromide

Bromide

SCHEMBL15775462

Br.N#Cc1cccc(C2=NC(=O)c3cccc(N)c3C2)c1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRA2C known ✓ P18825 1/20 0.38
XDH P47989 1/20 0.41
MAOB P27338 1/20 0.40
IDO1 P14902 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL15775523 0.88 LAP3 (0.40) MAOBIDO1
SCHEMBL15775980 0.86 LAP3 (0.41) MAOBIDO1
Bromide SCHEMBL15775614 0.81 GRM2 (0.40) MAOBIDO1
SCHEMBL15775665 0.80 ALDH1A1 (0.40)
Bromide SCHEMBL15775416 0.78 ADORA1 (0.43) MAOBIDO1
Bromide SCHEMBL15775859 0.78 XDH (0.41) XDHMAOB
Bromide SCHEMBL15775833 0.76 RXFP1 (0.34) MAOBCLK4
Bromide SCHEMBL15775323 0.76 TYR (0.41) MAOB
SCHEMBL15775366 0.74 RAB9A (0.38)
Bromide SCHEMBL15776793 0.74 BCHE (0.35) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed