SCHEMBL159204

SCHEMBL159204

O=C(ON1C(=O)CCC1=O)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
MGLL Q99685 3/20 0.41
FAAH O00519 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 5/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
MAPK1 P28482 2/20 0.40
HTT P42858 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
TP53 P04637 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HSD17B10 Q99714 1/20 0.39
ATM Q13315 1/20 0.39
PKM P14618 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1696262 1.00 KDM4E (0.42) KDM4ECES2CES1MGLLFAAH
SCHEMBL300884 0.91 CA12 (0.42) KDM4EMGLLMEN1KMT2AMAPT
SCHEMBL18119790 0.90 KDM4E (0.39) KDM4ECES2CES1MGLLFAAH
SCHEMBL13455758 0.85 SMN1; SMN2 (0.44) KDM4EMGLLMEN1KMT2ARAB9A
SCHEMBL5648489 0.84 CA12 (0.47) MEN1KMT2AMAPTRAB9AMAPK1
SCHEMBL27717830 0.84 CA1 (0.55) MGLLKMT2AMAPTHTTCA1
SCHEMBL1800956 0.82 PTPRF (0.44) KDM4ECES2CES1MAPTNPC1
SCHEMBL10070313 0.82 ALDH1A1 (0.37) KDM4EMGLLMEN1KMT2AMAPT
SCHEMBL16005095 0.82 ALDH1A1 (0.37) KDM4EMGLLMEN1KMT2AMAPT
SCHEMBL12216547 0.82 LMNA (0.44) KMT2AMAPTNPC1RAB9ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 171 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116761810-A Imaging and targeting of programmed death ligand-1 (PD-L1) expression 约翰霍普金斯大学 2023-09-15 CN claimed
US-20230271923-A1 IMAGING AND TARGETING PROGRAMMED DEATH LIGAND-1 (PD-LI) EXPRESSION THE JOHNS HOPKINS UNIVERSTY 2023-08-31 US claimed
CN-112675311-B 18/19 F-labeled PSMA (PSMA-conjugated diene monomer) targeting diagnosis and treatment integrated small-molecule drug conjugate, and preparation method and application thereof 西安交通大学医学院第一附属医院 2023-06-20 CN claimed
EP-4192524-A2 IMAGING AND TARGETING PROGRAMMED DEATH LIGAND-1 (PD-LI) EXPRESSION The Johns Hopkins University (US) 2023-06-14 EP claimed
US-11607466-B2 Tumor and immune cell imaging based on PD-L1 expression THE JOHNS HOPKINS UNIVERSITY (US) 2023-03-21 US claimed
WO-2022032100-A2 IMAGING AND TARGETING PROGRAMMED DEATH LIGAND-1 (PD-LI) EXPRESSION THE JOHNS HOPKINS UNIVERSITY (US) 2022-02-10 WO claimed
CN-112675311-A 18/19F-labeled PSMA (patterned beam-selective membrane array) targeted diagnosis and treatment integrated small-molecule drug conjugate, and preparation method and application thereof 西安交通大学医学院第一附属医院 2021-04-20 CN claimed
EP-3558395-A1 TUMOR AND IMMUNE CELL IMAGING BASED ON PD-L1 EXPRESSION The Johns Hopkins University (US) 2019-10-30 EP claimed
CN-110366432-A Tumour and immunocyte imaging based on PD-L1 expression 约翰霍普金斯大学 2019-10-22 CN claimed
US-20190314531-A1 TUMOR AND IMMUNE CELL IMAGING BASED ON PD-L1 EXPRESSION THE JOHNS HOPKINS UNIVERSITY 2019-10-17 US claimed
WO-2018119313-A1 TUMOR AND IMMUNE CELL IMAGING BASED ON PD-L1 EXPRESSION THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-28 WO claimed
US-12583913-B2 Antibody specific to Staphylococcus aureus, therapeutic method and detection method using same CHURCH WILLIAM R (US) 2026-03-24 US disclosed
US-20250375542-A1 18F-LABELED PSMA-TARGETED PET IMAGING AGENTS CANCER TARGETED TECH LLC (US) 2025-12-11 US disclosed
US-20250163104-A1 MACROCYCLIC IMMUNOMODULATORS BRISTOL MYERS SQUIBB CO (US) 2025-05-22 US disclosed
US-12139470-B2 Trioxolane agents THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-11-12 US disclosed
WO-2006032911-A2 METALLOPROTEINASE INHIBITOR IMAGING AGENTS GE HEALTHCARE LIMITED (GB) 2006-03-30 WO disclosed
EP-1142890-B1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG CO LTD (JP) 2005-08-03 EP disclosed
US-6511997-B1 For treatment of a disease associated with tumor necrosis factor alpha, interleukin 1, interleukin 6 or cyclooxygenase II; such as irritable bowel disease TEIKOKU HORMONE MFG. CO., LTD. (JP) 2003-01-28 US disclosed
CN-1331688-A Aminopyridine Derivatives TEIKOKU HORMONE MFG CO LTD (JP) 2002-01-16 CN disclosed
EP-1142890-A1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG. CO., LTD. (JP) 2001-10-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12139470-B2 Trioxolane agents ABCB4, SLC10A1, SLC10A2 KDM4E 4796/4885CES2 2373/4885CES1 330/4885
US-20250163104-A1 MACROCYCLIC IMMUNOMODULATORS CD274, PDCD1LG2, PDCD1 KDM4E 1355/4885CES2 4750/4885CES1 4282/4885
US-12583913-B2 Antibody specific to Staphylococcus aureus, therapeutic method and detection method using same IGSF11, VSIG8, VARS1 KDM4E 1665/4885CES2 3583/4885CES1 1997/4885
US-11607466-B2 Tumor and immune cell imaging based on PD-L1 expression CD274, PDCD1LG2, PDCD1 KDM4E 4444/4885CES2 4488/4885CES1 2996/4885
US-20190314531-A1 TUMOR AND IMMUNE CELL IMAGING BASED ON PD-L1 EXPRESSION CD274, PDCD1LG2, PDCD1 KDM4E 4444/4885CES2 4488/4885CES1 2996/4885
US-20230271923-A1 IMAGING AND TARGETING PROGRAMMED DEATH LIGAND-1 (PD-LI) EXPRESSION CD274, PDCD1LG2, PDCD1 KDM4E 4400/4885CES2 4548/4885CES1 4149/4885
US-20250375542-A1 18F-LABELED PSMA-TARGETED PET IMAGING AGENTS FOLH1, PSMA1, PSMA2 KDM4E 2380/4885CES2 1560/4885CES1 966/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.