SCHEMBL15925898

SCHEMBL15925898

NC1=N[C@@H](CCc2ccc(F)cc2F)CCC1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 11/20 0.48
NOS2 P35228 10/20 0.48
NOS3 P29474 7/20 0.48
HTR2A P28223 5/20 0.43
HTR2C P28335 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925910 0.78 NOS1 (0.54) NOS1NOS2NOS3
SCHEMBL3607332 0.74
SCHEMBL3607329 0.74
SCHEMBL16191075 0.73 HTR2A (0.58) HTR2AHTR2C
SCHEMBL8202601 0.71 LOXL2 (0.45) NOS1NOS2NOS3
SCHEMBL8200215 0.71 NOS1 (0.46) NOS1NOS2NOS3
SCHEMBL8153366 0.68 HTR2A (0.56) HTR2AHTR2C
SCHEMBL8147279 0.68 HTR2A (0.56) HTR2AHTR2C
SCHEMBL8148467 0.68 HTR2A (0.56) HTR2AHTR2C
SCHEMBL22201819 0.68 HTR2A (0.52) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114906-B1 2-AMINOOXAZOLINES AS TAAR1 LIGANDS FOR CNS DISORDERS HOFFMANN LA ROCHE (CH) 2014-08-06 EP disclosed