SCHEMBL15933683

SCHEMBL15933683

CC(C)(C)OC(=O)N1CCn2nc(-c3cncc(C#N)c3)nc2C1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.52
EGLN2 Q96KS0 1/20 0.39
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
CYP11B2 P19099 2/20 0.37
CYP11B1 P15538 1/20 0.37
ESR2 Q92731 1/20 0.36
GBA1 P04062 1/20 0.36
PGGT1B P53609 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
CETP P11597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933535 0.87 GPR119 (0.49) GPR119EGLN2ESR2PGGT1BCETP
SCHEMBL15933678 0.86 CSNK1D (0.43) GPR119ESR2GBA1
SCHEMBL15933643 0.84 GPR119 (0.45) GPR119ESR2GBA1
SCHEMBL15933677 0.81 GPR119 (0.53) GPR119EGLN2BRD4CREBBP
SCHEMBL15933697 0.80 GPR119 (0.47) GPR119ESR2GBA1
SCHEMBL17984905 0.79 ESR2 (0.40) ESR2
SCHEMBL20140942 0.79 CKS1B (0.49) GPR119ESR2GBA1
SCHEMBL25431827 0.77 GPR119 (0.43) GPR119ESR2
SCHEMBL24689592 0.76 PDE10A (0.42) GPR119GBA1
SCHEMBL15933477 0.76 HDAC4 (0.40) GPR119ESR2GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed