SCHEMBL15960708

SCHEMBL15960708

CC(C)N1CCC2(CCCO2)C1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.33
KCNH2 Q12809 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15960715 0.94 KCNH2 (0.36) RORCKCNH2CYP2D6
SCHEMBL9963383 0.92 RORC (0.31) RORC
SCHEMBL27380449 0.90 CYP2D6 (0.33) CYP2D6
SCHEMBL15960718 0.90 CYP2D6 (0.33) CYP2D6
SCHEMBL25081767 0.89
SCHEMBL9963298 0.88 CYP2D6 (0.36) KCNH2CYP2D6CYP11B1CYP11B2
SCHEMBL9963384 0.87 KCNH2 (0.33) KCNH2
SCHEMBL17014689 0.86 MGLL (0.30)
SCHEMBL25081715 0.86
SCHEMBL9963380 0.86 HRH3 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239813-A1 KRAS INHIBITORS AND PHARMACEUTICAL USES THEREOF Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2024-07-18 US disclosed
US-20240239813-A1 KRAS INHIBITORS AND PHARMACEUTICAL USES THEREOF Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2024-07-18 US disclosed
US-20240217952-A1 TREATMENT OF GRAFT-VERSUS-HOST DISEASE WITH INHIBITORS OF BET FAMILY BDII BROMODOMAIN POSEIDON INNOVATION 1, INC. 2024-07-04 US disclosed
US-20240217952-A1 TREATMENT OF GRAFT-VERSUS-HOST DISEASE WITH INHIBITORS OF BET FAMILY BDII BROMODOMAIN POSEIDON INNOVATION 1, INC. 2024-07-04 US disclosed
US-20240025918-A1 KRAS G12D Inhibitors JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-01-25 US disclosed
US-20240025918-A1 KRAS G12D Inhibitors JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-01-25 US disclosed
WO-2023247593-A1 PYRROLOPYRIDINE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2023-12-28 WO disclosed
US-11834455-B2 Carm1 inhibitors and uses thereof Epizyme, Inc. (US) 2023-12-05 US disclosed
US-20230279020-A9 CARM1 INHIBITORS AND USES THEREOF Epizyme, Inc. (US) 2023-09-07 US disclosed
US-20230112485-A1 THERAPEUTIC COMPOUNDS GENENTECH, INC. (US) 2023-04-13 US disclosed
US-20160237093-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA BIO, Inc. 2016-08-18 US disclosed
US-20160235761-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA BIO, Inc. 2016-08-18 US disclosed
US-20160235753-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA BIO, Inc. 2016-08-18 US disclosed
US-20160237094-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA BIO, Inc. 2016-08-18 US disclosed
US-9353123-B2 Therapeutic compounds and uses thereof KALA PHARMACEUTICALS, INC. (US) 2016-05-31 US disclosed
US-9353122-B2 Therapeutic compounds and uses thereof KALA PHARMACEUTICALS, INC. (US) 2016-05-31 US disclosed
US-20160039834-A1 CARM1 INHIBITORS AND USES THEREOF Epizyme, Inc. (US) 2016-02-11 US disclosed
US-20160002254-A1 Therapeutic Compounds and Uses Thereof KALA PHARMACEUTICALS, INC. (US) 2016-01-07 US disclosed
US-20140235634-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA PHARMACEUTICALS, INC. (US) 2014-08-21 US disclosed
US-20140235657-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF KALA PHARMACEUTICALS, INC. (US) 2014-08-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (14 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230112485-A1 THERAPEUTIC COMPOUNDS BRDT, BRPF3, SNRPE RORC 2184/4885KCNH2 4724/4885CYP2D6 4859/4885
US-20140235657-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 627/4885KCNH2 3015/4885CYP2D6 1098/4885
US-20230279020-A9 CARM1 INHIBITORS AND USES THEREOF CARM1, TIAM1, ADRM1 RORC 371/4885KCNH2 4678/4885CYP2D6 1700/4885
US-20160235753-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 627/4885KCNH2 3015/4885CYP2D6 1098/4885
US-11834455-B2 Carm1 inhibitors and uses thereof CARM1, TIAM1, ADRM1 RORC 360/4885KCNH2 4676/4885CYP2D6 1699/4885
US-20240217952-A1 TREATMENT OF GRAFT-VERSUS-HOST DISEASE WITH INHIBITORS OF BET FAMILY BDII BROMODOMAIN BRDT, BET1, BRD4 RORC 1045/4885KCNH2 4663/4885CYP2D6 4337/4885
US-20160235761-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 516/4885KCNH2 3314/4885CYP2D6 419/4885
US-20160237094-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 627/4885KCNH2 3015/4885CYP2D6 1098/4885
US-20160237093-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 516/4885KCNH2 3314/4885CYP2D6 419/4885
US-20240239813-A1 KRAS INHIBITORS AND PHARMACEUTICAL USES THEREOF KRAS, NRAS, HRAS RORC 1334/4885KCNH2 4693/4885CYP2D6 2058/4885
US-20140235634-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF MUC1, CFTR, SLC26A4 RORC 516/4885KCNH2 3314/4885CYP2D6 419/4885
US-20160002254-A1 Therapeutic Compounds and Uses Thereof PCSK9, CFTR, SLC10A1 RORC 146/4885KCNH2 3197/4885CYP2D6 256/4885
US-20240025918-A1 KRAS G12D Inhibitors KRAS, NRAS, HRAS RORC 317/4885KCNH2 4548/4885CYP2D6 2836/4885
US-20160039834-A1 CARM1 INHIBITORS AND USES THEREOF CARM1, TIAM1, ADRM1 RORC 393/4885KCNH2 4671/4885CYP2D6 1709/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.