SCHEMBL15966849

SCHEMBL15966849

CSC1C(=O)Nc2c(F)cccc21.O=C1Cc2cccc(F)c2N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.41
SMYD3 Q9H7B4 2/20 0.34
SRD5A1 P18405 1/20 0.33
HTR5A P47898 1/20 0.33
OPRL1 P41146 1/20 0.33
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
PDK2 Q15119 1/20 0.33
TP53 P04637 1/20 0.32
TDP2 O95551 2/20 0.31
CASP3 P42574 1/20 0.31
CASP7 P55210 1/20 0.31
CASP9 P55211 1/20 0.31
CASP6 P55212 1/20 0.31
CASP8 Q14790 1/20 0.31
MAP3K14 Q99558 1/20 0.31
GRM5 P41594 1/20 0.31
ALDH1A1 P00352 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL116597 0.87 ALDH1A1 (0.37) PDK2TP53ALDH1A1DDB1CRBN
SCHEMBL15966870 0.82 AHR (0.62) AHRSMYD3HTR5AGRIA1CACNG8
SCHEMBL15966884 0.81 HTR5A (0.40) AHRSMYD3HTR5ATP53ALDH1A1
SCHEMBL261018 0.79 AHR (0.61) AHRSMYD3SRD5A1HTR5AOPRL1
SCHEMBL15967351 0.78 GRIA1 (0.33) GRIA1CACNG8TDP2
SCHEMBL10952280 0.71 ALDH1A1 (0.37) ALDH1A1
SCHEMBL11368672 0.70 DAO (0.40) PDK2ALDH1A1DDB1CRBN
SCHEMBL117727 0.69 CACNB4 (0.40) AHRCACNG8ALDH1A1
SCHEMBL11094086 0.68 HTR1A (0.34) HTR5AALDH1A1
SCHEMBL1321330 0.67 HTR2C (0.46) HTR5AALDH1A1DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569283-B1 METHOD FOR PRODUCING SUBSTITUTED 1,3-DIHYDRO-2H-INDOL-2-ONES BAYER IP GMBH (DE) 2014-08-27 EP disclosed