SCHEMBL16004143

SCHEMBL16004143

O=C(c1cccs1)N1CCOc2ccc(COCc3cccc(F)c3)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
GPR142 Q7Z601 2/20 0.43
RIPK1 Q13546 1/20 0.43
GAA P10253 4/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KCNA5 P22460 1/20 0.38
PIK3CA P42336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004095 0.85 LMNA (0.43) LMNARIPK1GAAKDM4EALDH1A1
SCHEMBL16004103 0.84 LMNA (0.44) LMNAGAAALDH1A1CYP2C9HTT
SCHEMBL16004140 0.84 LMNA (0.44) LMNAGPR142RIPK1GAAALDH1A1
SCHEMBL16003974 0.83 HRH3 (0.52) LMNAGAAKCNA5
SCHEMBL16003983 0.83 GAA (0.43) LMNARIPK1GAAALDH1A1CYP2C9
SCHEMBL16003973 0.83 TSHR (0.46) GPR142RIPK1KDM4EALDH1A1HTT
SCHEMBL16004139 0.80 ALDH1A1 (0.53) LMNAGPR142RIPK1KDM4EALDH1A1
SCHEMBL16003982 0.80 ALDH1A1 (0.45) GPR142RIPK1KDM4EALDH1A1HTT
SCHEMBL16004295 0.80 RIPK1 (0.44) GPR142RIPK1KDM4EALDH1A1HTT
SCHEMBL16004094 0.80 GPR142 (0.64) GPR142

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed