SCHEMBL16004139

SCHEMBL16004139

COc1cccc(C(=O)N2CCOc3ccc(COCc4cccc(F)c4)cc3C2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
KMT2A Q03164 3/20 0.53
KDM4E B2RXH2 2/20 0.53
MEN1 O00255 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.49
HTT P42858 2/20 0.45
GPR142 Q7Z601 2/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HSD11B1 P28845 1/20 0.43
RIPK1 Q13546 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16003982 0.87 ALDH1A1 (0.45) ALDH1A1KMT2AKDM4EL3MBTL1HTT
SCHEMBL16004136 0.85 GPR142 (0.46) ALDH1A1KMT2ASMN1; SMN2L3MBTL1GPR142
SCHEMBL16004302 0.83 ALDH1A1 (0.51) ALDH1A1KMT2ASMN1; SMN2L3MBTL1HTT
SCHEMBL16004298 0.83 ALDH1A1 (0.49) ALDH1A1KDM4ESMN1; SMN2HTTGPR142
SCHEMBL16003973 0.81 TSHR (0.46) ALDH1A1KMT2AKDM4EMEN1SMN1; SMN2
SCHEMBL16003972 0.81 HSD11B1 (0.45) ALDH1A1L3MBTL1GPR142HSD11B1RIPK1
SCHEMBL16004143 0.80 LMNA (0.43) ALDH1A1KDM4ESMN1; SMN2HTTGPR142
SCHEMBL16003978 0.80 L3MBTL1 (0.45) ALDH1A1KMT2AMEN1SMN1; SMN2L3MBTL1
SCHEMBL16004311 0.80 GPR142 (0.64) ALDH1A1HTTGPR142NPC1RAB9A
SCHEMBL16004138 0.79 SIGMAR1 (0.48) KMT2AMEN1GPR142NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed