SCHEMBL16004243

SCHEMBL16004243

CCC(=O)N(C)Cc1ccc2c(c1)CN(C(=O)c1ccsc1)CCO2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.40
RIPK1 Q13546 3/20 0.40
AOC3 Q16853 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.36
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004271 0.84 RIPK1 (0.45) PIK3CARIPK1AOC3MEN1KMT2A
SCHEMBL16004232 0.83 PIK3CA (0.49) PIK3CARIPK1AOC3HPGD
SCHEMBL16004283 0.81 CREBBP (0.52) CREBBP
SCHEMBL16004052 0.78 PIK3CA (0.52) PIK3CARIPK1AOC3HPGD
SCHEMBL16004055 0.77 PIK3CA (0.49) PIK3CARIPK1MEN1KMT2A
SCHEMBL16004054 0.77 PIK3CA (0.49) PIK3CARIPK1AOC3MEN1KMT2A
SCHEMBL16004274 0.77 RIPK1 (0.46) PIK3CARIPK1MEN1KMT2AHPGD
SCHEMBL16004053 0.77 RIPK1 (0.49) PIK3CARIPK1
SCHEMBL16004269 0.75 RIPK1 (0.46) PIK3CARIPK1MEN1KMT2AHPGD
SCHEMBL16004059 0.75 HPGD (0.47) PIK3CAKMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed