SCHEMBL16004271

SCHEMBL16004271

CCC(=O)N(C)Cc1ccc2c(c1)CN(C(C)=O)CCO2

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.45
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NTRK1 P04629 1/20 0.40
PIK3CA P42336 4/20 0.39
CREBBP Q92793 4/20 0.38
AOC3 Q16853 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
GPR142 Q7Z601 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004269 0.91 RIPK1 (0.46) RIPK1MEN1KMT2ANTRK1PIK3CA
SCHEMBL16004283 0.88 CREBBP (0.52) CREBBP
SCHEMBL16004274 0.85 RIPK1 (0.46) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004243 0.84 PIK3CA (0.40) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004232 0.82 PIK3CA (0.49) RIPK1PIK3CAAOC3GAAHPGD
SCHEMBL16004285 0.80 CREBBP (0.54) CREBBP
SCHEMBL16004236 0.80 KDM4E (0.43) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004249 0.78 RIPK1 (0.41) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004052 0.78 PIK3CA (0.52) RIPK1PIK3CAAOC3ALDH1A1GAA
SCHEMBL16004055 0.78 PIK3CA (0.49) RIPK1MEN1KMT2APIK3CAGPR142

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed