SCHEMBL16004269

SCHEMBL16004269

CC(=O)N(C)Cc1ccc2c(c1)CN(C(C)=O)CCO2

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.46
NTRK1 P04629 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PIK3CA P42336 3/20 0.41
CREBBP Q92793 4/20 0.40
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
DGAT1 O75907 1/20 0.38
GPR142 Q7Z601 2/20 0.38
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004271 0.91 RIPK1 (0.45) RIPK1NTRK1MEN1KMT2APIK3CA
SCHEMBL16004274 0.90 RIPK1 (0.46) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004285 0.89 CREBBP (0.54) CREBBP
SCHEMBL16004236 0.89 KDM4E (0.43) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004052 0.87 PIK3CA (0.52) RIPK1PIK3CAALDH1A1GAAHPGD
SCHEMBL16004249 0.87 RIPK1 (0.41) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004054 0.86 PIK3CA (0.49) RIPK1MEN1KMT2APIK3CACREBBP
SCHEMBL16004233 0.86 GPR142 (0.47) RIPK1KMT2APIK3CAALDH1A1GAA
SCHEMBL16004055 0.86 PIK3CA (0.49) RIPK1MEN1KMT2APIK3CAGPR142
SCHEMBL16004053 0.85 RIPK1 (0.49) RIPK1PIK3CAALDH1A1GAAGPR142

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed