SCHEMBL16004274

SCHEMBL16004274

CCC(=O)N1CCOc2ccc(CN(C)C(C)=O)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.46
CREBBP Q92793 4/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GPR142 Q7Z601 2/20 0.39
PIK3CA P42336 4/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
DGAT1 O75907 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004236 0.90 KDM4E (0.43) RIPK1CREBBPMEN1KMT2AGPR142
SCHEMBL16004269 0.90 RIPK1 (0.46) RIPK1CREBBPMEN1KMT2AGPR142
SCHEMBL16004249 0.88 RIPK1 (0.41) RIPK1CREBBPMEN1KMT2AGPR142
SCHEMBL16004233 0.87 GPR142 (0.47) RIPK1KMT2AGPR142PIK3CAMAPT
SCHEMBL16004271 0.85 RIPK1 (0.45) RIPK1CREBBPMEN1KMT2AGPR142
SCHEMBL16004285 0.85 CREBBP (0.54) CREBBP
SCHEMBL16004052 0.84 PIK3CA (0.52) RIPK1PIK3CAALDH1A1HPGDGAA
SCHEMBL16004054 0.83 PIK3CA (0.49) RIPK1CREBBPMEN1KMT2APIK3CA
SCHEMBL16004055 0.83 PIK3CA (0.49) RIPK1MEN1KMT2AGPR142PIK3CA
SCHEMBL16004053 0.82 RIPK1 (0.49) RIPK1GPR142PIK3CAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed