Levopropylhexedrine

Levopropylhexedrine

SCHEMBL161851

CN[C@@H](C)CC1CCCCC1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.42
SIGMAR1 Q99720 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CTSL P07711 3/20 0.35
CTSB P07858 3/20 0.35
CTSH P09668 2/20 0.35
LTA4H P09960 1/20 0.35
CYP1A2 P05177 1/20 0.34
METAP2 P50579 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levopropylhexedrine SCHEMBL20780004 1.00 CTSK (0.42) CTSKSIGMAR1MEN1KMT2ACTSL
Propylhexedrine SCHEMBL28537 1.00 CTSK (0.42) CTSKSIGMAR1MEN1KMT2ACTSL
Propylhexedrine SCHEMBL28890426 0.98 CTSK (0.41) CTSKSIGMAR1MEN1KMT2ACTSL
Propylhexedrine SCHEMBL4900116 0.98 CTSK (0.41) CTSKSIGMAR1MEN1KMT2ACTSL
Cyclopentamine SCHEMBL13479599 0.98 CTSK (0.40) CTSKSIGMAR1MEN1KMT2ACTSL
Cyclopentamine SCHEMBL249708 0.98 CTSK (0.40) CTSKSIGMAR1MEN1KMT2ACTSL
Cyclopentamine SCHEMBL317336 0.95 CTSK (0.39) CTSKSIGMAR1MEN1KMT2ACTSL
SCHEMBL27308544 0.93
SCHEMBL22627190 0.81 CTSK (0.32) CTSK
SCHEMBL23241391 0.79 OPRK1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 143 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240226084-A9 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS TECHFIELDS PHARMA CO., LTD. (CN) 2024-07-11 US claimed
US-20240131017-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS TECHFIELDS PHARMA CO., LTD. (CN) 2024-04-25 US claimed
US-20240115562-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS TECHFIELDS PHARMA CO., LTD. (CN) 2024-04-11 US claimed
US-20200060997-A1 TARR Receptor Agonists for Sexual Dysfunction JOHN MCCOY 2020-02-27 US claimed
EP-3366306-A2 USE OF SOME PEPTIDES IN DIAGNOSIS AND TREATMENT OF DIABETES, OBESITY AND METABOLIC DISEASES ASSOCIATED THERETO Istanbul Universitesi Rektorlugu (TR) 2018-08-29 EP claimed
EP-3351262-A1 CURAGLUTIDE FOR IN TREATMENT OF PREDIABETES, DIABETES, OBESITY AND METABOLIC DISEASES ASSOCIATED THERETO Istanbul Universitesi Rektorlugu (TR) 2018-07-25 EP claimed
US-20150072961-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS PREMIER RESEARCH INTERNATIONAL, LLC 2015-03-12 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1497272-A4 METHOD OF PREPARING AMINE STEREOISOMERS APSINTERM LLC (US) 2007-02-07 EP claimed
US-7129378-B2 Method of preparing amine stereoisomers APSINTERM, LLC (US) 2006-10-31 US claimed
US-20050165240-A1 Method of preparing amine stereoisomers APSINTERM, LLC 2005-07-28 US claimed
EP-1497272-A2 METHOD OF PREPARING AMINE STEREOISOMERS Apsinterm, LLC. (US) 2005-01-19 EP claimed
WO-2003091207-A2 METHOD OF PREPARING AMINE STEREOISOMERS APSINTERM, LLC. (US) 2003-11-06 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2026106796-A1 SYSTEM AND METHOD FOR THE TREATMENT OF TELOGEN EFFLUVIUM, ANDROGENETIC ALOPECIA, AND OTHER HAIR LOSS DISORDERS FOLLEA INTERNATIONAL (US) 2026-05-21 WO disclosed
US-20260041652-A1 SYSTEM AND METHOD FOR PREVENTING ALOPECIA FOLLEA INT (US) 2026-02-12 US disclosed
EP-4079311-B1 NMN AND DERIVATIVES FOR USE IN THE TREATMENT OF DEPRESSION AND/OR ANXIETY IN PATIENTS HAVING A FORM OF PARKINSONISM NUVAMID SA (CH) 2025-10-01 EP disclosed
US-6288040-B1 CARRIER SURFACE BONDED TO RECOGNITION PROTEINS; DRUG DELIVERY; CENTRAL NERVOUS SYSTEM DISORDERS DSS DRUG DELIVERY SERVICE GESELLSCHAFT ZUR FORDERUNG DER FOSHUNG IN PHAMAZEUTISCHER TECHNOLOGI UND BIOPHARMAZIE MBH (DE) 2001-09-11 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240226084-A9 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS HRH4, HCAR2, PAH CTSK 736/4885SIGMAR1 3110/4885MEN1 2172/4885
US-20050165240-A1 Method of preparing amine stereoisomers SRM, TST, SMOX CTSK 4526/4885SIGMAR1 411/4885MEN1 2372/4885
US-20240115562-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS HRH4, HCAR2, PAH CTSK 736/4885SIGMAR1 3110/4885MEN1 2172/4885
US-20150072961-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS HRH4, HCAR2, PAH CTSK 736/4885SIGMAR1 3110/4885MEN1 2172/4885
US-20240131017-A1 HIGH PENETRATION PRODRUG COMPOSITIONS AND PHARMACEUTICAL COMPOSITION THEREOF FOR TREATMENT OF PULMONARY CONDITIONS HRH4, HCAR2, PAH CTSK 736/4885SIGMAR1 3110/4885MEN1 2172/4885
US-20260041652-A1 SYSTEM AND METHOD FOR PREVENTING ALOPECIA DYRK4, DYRK2, STRA6 CTSK 1429/4885SIGMAR1 4868/4885MEN1 4129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.