SCHEMBL16200062

SCHEMBL16200062

COc1ccc(-c2nn(C)c(C(F)(F)F)c2Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.46
PTGS1 P23219 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
THPO P40225 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
HIF1A Q16665 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 3/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12859380 0.87 MEN1 (0.40) PTGS2NPSR1KDM4EALDH1A1RAB9A
SCHEMBL16200053 0.83 SLC34A1 (0.44) PTGS2PTGS1RAB9ASMN1; SMN2MAPT
SCHEMBL14039900 0.81 ALDH1A1 (0.50) CYP1A2CYP2C9CYP2C19NPSR1KDM4E
SCHEMBL16200057 0.80 MAPK14 (0.42) CYP1A2CYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL14996631 0.78 MEN1 (0.43) PTGS2NPSR1KDM4EALDH1A1RAB9A
SCHEMBL8108697 0.77 SLC34A1 (0.38) CYP1A2CYP2C9CYP2C19NPSR1KDM4E
SCHEMBL13739115 0.75 ALDH1A1 (0.55) NPSR1KDM4EALDH1A1RAB9ANPC1
SCHEMBL8475975 0.74 F2RL3 (0.38) PTGS2NPSR1KDM4EALDH1A1RAB9A
SCHEMBL7780377 0.74 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL14039556 0.73 NT5E (0.41) PTGS2CYP1A2CYP3A4TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed