SCHEMBL16200063

SCHEMBL16200063

Cc1c(Cl)c(-c2cccnc2)nn1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
CYP2A6 P11509 7/20 0.47
CYP2A13 Q16696 1/20 0.46
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
P2RX7 Q99572 1/20 0.42
NPY5R Q15761 2/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2B6 P20813 1/20 0.41
MAP2K4 P45985 1/20 0.40
CYP11B2 P19099 1/20 0.40
TBXAS1 P24557 1/20 0.40
HK1 P19367 1/20 0.40
HKDC1 Q2TB90 1/20 0.40
CYP2D6 P10635 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19453173 0.83 CYP2A6 (0.50) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL2690242 0.83 CYP2A6 (0.45) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL2690686 0.81 CYP2A6 (0.44) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL16200060 0.81 THRB (0.52) ALDH1A1CYP1A2THRBCYP2C9CYP2C19
SCHEMBL16200054 0.79 P2RX7 (0.45) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL2690682 0.79 CYP2A6 (0.43) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL13184419 0.79 PTGS2 (0.39) ALDH1A1THRB
SCHEMBL16200083 0.77 ALDH1A1 (0.48) ALDH1A1CYP2A6CYP2A13CYP1A2CYP3A4
SCHEMBL16200199 0.75 MEN1 (0.43) ALDH1A1CYP2A6THRB
SCHEMBL14996629 0.74 NR1H2 (0.44) ALDH1A1CYP1A2THRBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed