SCHEMBL16200323

SCHEMBL16200323

Cc1c(Cl)c(-c2cn[nH]c2)nn1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
THRB P10828 1/20 0.39
GFER P55789 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
KDM4E B2RXH2 1/20 0.36
KCNH2 Q12809 1/20 0.35
AKT1 P31749 2/20 0.35
AKT2 P31751 1/20 0.35
PDE10A Q9Y233 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15716268 0.73 MTOR (0.38) ALDH1A1GAALMNAMAPTKDM4E
SCHEMBL25753038 0.72 BRD4 (0.39) LMNAMAPTKCNH2AKT1AKT2
SCHEMBL14996558 0.72 ALDH1A1 (0.52) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL14996629 0.72 NR1H2 (0.44) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL16200060 0.72 THRB (0.52) ALDH1A1GAAHPGDTHRBNPSR1
SCHEMBL16200055 0.70 MAPK14 (0.43) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL14996631 0.70 MEN1 (0.43) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL13184419 0.70 PTGS2 (0.39) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL16200199 0.70 MEN1 (0.43) ALDH1A1GAAHPGDTHRBGFER
SCHEMBL21241065 0.69 PIM1 (0.42) ALDH1A1LMNAAPOBEC3GKDM4EKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed