SCHEMBL16227684

SCHEMBL16227684

NCCSSCCNC(=O)CCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.43
KDM4E B2RXH2 3/20 0.42
KDM5C P41229 3/20 0.42
PHF8 Q9UPP1 3/20 0.42
KDM2A Q9Y2K7 3/20 0.42
EGLN1 Q9GZT9 2/20 0.39
KDM6B O15054 1/20 0.39
FOLH1 Q04609 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
ECE1 P42892 1/20 0.37
THPO P40225 1/20 0.37
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
EHMT2 Q96KQ7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GABRR1 P24046 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL23355106 0.91 TSHR (0.35) TSHRKDM4EKDM5CPHF8KDM2A
SCHEMBL24329788 0.90 TSHR (0.52) TSHRKDM4EKDM5CPHF8KDM2A
SCHEMBL13340981 0.84 PAOX (0.37) TSHRKDM4ECA1CA2CA9
Alethine SCHEMBL689905 0.82 TSHR (0.41) TSHRCA1CA2CA9LMNA
Cystamine SCHEMBL28779847 0.82 TSHR (0.63) TSHRKDM4EKDM5CPHF8KDM2A
SCHEMBL18629861 0.81 TSHR (0.43) TSHRKDM4EKDM5CPHF8KDM2A
SCHEMBL14547392 0.81 CASP2 (0.48) TSHRTHPOLMNAALDH1A1HDAC3
SCHEMBL8582768 0.80 TSHR (0.43) TSHRCA1CA2CA9THPO
SCHEMBL766363 0.80 PHF8 (0.52) TSHRKDM4EKDM5CPHF8KDM2A
SCHEMBL16549625 0.79 FAAH (0.45) TSHRCA1CA2CA9THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112672747-B Peptides for activating cell signaling in osteoprogenitor cells 加利福尼亚大学董事会 2025-02-18 CN disclosed
CN-112703185-B Thiocycloheptyne derivatives and uses thereof 克里斯特递送有限公司 2024-12-27 CN disclosed
US-12157778-B2 Peptides for activation of cell signaling in osteoprogenitor cells THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-12-03 US disclosed
US-20210395216-A1 THIOCYCLOHEPTYNE DERIVATIVES AND THEIR USE CRISTAL DELIVERY B.V. (NL) 2021-12-23 US disclosed
US-20210395302-A1 PEPTIDES FOR ACTIVATION OF CELL SIGNALING IN OSTEOPROGENITOR CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-12-23 US disclosed
EP-3823630-A1 PEPTIDES FOR ACTIVATION OF CELL SIGNALING IN OSTEOPROGENITOR CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-05-26 EP disclosed
CN-112703185-A Thiocycloyne derivatives and uses thereof 克里斯特递送有限公司 2021-04-23 CN disclosed
CN-112672747-A Peptides for activating cell signalling in osteoprogenitor cells 加利福尼亚大学董事会 2021-04-16 CN disclosed
WO-2020013696-A9 THIOCYCLOHEPTYNE DERIVATIVES AND THEIR USE CRISTAL DELIVERY B.V. (NL) 2021-02-25 WO disclosed
WO-2020018941-A1 PEPTIDES FOR ACTIVATION OF CELL SIGNALING IN OSTEOPROGENITOR CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-01-23 WO disclosed
US-10322180-B2 Pharmaceutical composition comprising modified hemoglobin-based therapeutic agent for cancer targeting treatment and diagnostic imaging VISION GLOBAL HOLDINGS LTD. (HK) 2019-06-18 US disclosed
EP-3001813-B1 PHARMACEUTICAL COMPOSITION COMPRISING MODIFIED HEMOGLOBIN- BASED THERAPEUTIC AGENT FOR CANCER TARGETING TREATMENT AND DIAGNOSTIC IMAGING VISION GLOBAL HOLDINGS LTD (CN) 2019-03-27 EP disclosed
US-20170266285-A1 PHARMACEUTICAL COMPOSITION COMPRISING MODIFIED HEMOGLOBIN-BASED THERAPEUTIC AGENT FOR CANCER TARGETING TREATMENT AND DIAGNOSTIC IMAGING VISION GLOBAL HOLDINGS LTD. (HK) 2017-09-21 US disclosed
US-9636404-B2 Pharmaceutical composition comprising modified hemoglobin-based therapeutic agent for cancer targeting treatment and diagnostic imaging VISION GLOBAL HOLDINGS LTD. (CN) 2017-05-02 US disclosed
EP-3001813-A1 PHARMACEUTICAL COMPOSITION COMPRISING MODIFIED HEMOGLOBIN- BASED THERAPEUTIC AGENT FOR CANCER TARGETING TREATMENT AND DIAGNOSTIC IMAGING Vision Global Holdings Ltd. (CN) 2016-04-06 EP disclosed
WO-2014186301-A1 PHARMACEUTICAL COMPOSITION COMPRISING MODIFIED HEMOGLOBIN- BASED THERAPEUTIC AGENT FOR CANCER TARGETING TREATMENT AND DIAGNOSTIC IMAGING VISION GLOBAL HOLDINGS LTD. (CN) 2014-11-20 WO disclosed
US-20140335018-A1 PHARMACEUTICAL COMPOSITION COMPRISING MODIFIED HEMOGLOBIN-BASED THERAPEUTIC AGENT FOR CANCER TARGETING TREATMENT AND DIAGNOSTIC IMAGING VISION GLOBAL HOLDINGS LTD. (HK) 2014-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210395216-A1 THIOCYCLOHEPTYNE DERIVATIVES AND THEIR USE CYP7A1, CYP3A5, ABCB1 TSHR 642/4885KDM4E 3076/4885KDM5C 1197/4885
US-20210395302-A1 PEPTIDES FOR ACTIVATION OF CELL SIGNALING IN OSTEOPROGENITOR CELLS ITGB4, ITGA4, ITGB1 TSHR 1563/4885KDM4E 2319/4885KDM5C 3261/4885
US-10322180-B2 Pharmaceutical composition comprising modified hemoglobin-based therapeutic agent for cancer targeting treatment and diagnostic imaging HBG2, HBG1, HBB TSHR 714/4885KDM4E 1846/4885KDM5C 875/4885
US-12157778-B2 Peptides for activation of cell signaling in osteoprogenitor cells ITGB4, ITGA4, ITGB1 TSHR 1563/4885KDM4E 2319/4885KDM5C 3261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.