SCHEMBL16229798

SCHEMBL16229798

CN1C2C1C21Cc2cc(F)c(CCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.36
SLC6A9 P48067 1/20 0.34
PKM P14618 1/20 0.34
AKR1C3 P42330 1/20 0.34
SLC8A1 P32418 1/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
TSHR P16473 2/20 0.33
TAAR1 Q96RJ0 2/20 0.33
GAA P10253 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPK1 P28482 1/20 0.33
LIPC P11150 1/20 0.32
MAPT P10636 1/20 0.32
EP300 Q09472 2/20 0.32
HTT P42858 1/20 0.32
HTR1A P08908 1/20 0.32
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229806 0.93 DGAT1 (0.35) HTR6SLC6A9AKR1C3ALDH1A1LMNA
SCHEMBL16784652 0.92 SLC8A1 (0.37) SLC6A9SLC8A1LMNAKDM4ELIPC
SCHEMBL16229761 0.92 SLC6A9 (0.37) HTR6SLC6A9AKR1C3ALDH1A1LMNA
SCHEMBL16229800 0.90 SLC6A9 (0.36) HTR6SLC6A9HTR1AHTR7
SCHEMBL16784640 0.88 SLC6A9 (0.41) HTR6SLC6A9SLC8A1ALDH1A1HTR1A
SCHEMBL16229746 0.87 HTT (0.40) SLC6A9PKMSLC8A1ALDH1A1LMNA
SCHEMBL16229792 0.85 POLB (0.35) SLC6A9PKMSLC8A1ALDH1A1KDM4E
SCHEMBL16229748 0.85 SLC6A9 (0.45) SLC6A9LMNAGAA
SCHEMBL16229766 0.84 TP53 (0.35) SLC6A9PKMSLC8A1MAPK1
SCHEMBL16229772 0.82 AXL (0.37) SLC6A9SLC8A1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed
US-8883839-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy ABBOTT LABORATORIES (US) 2014-11-11 US disclosed