SCHEMBL16239477

SCHEMBL16239477

CC1(C)CC(c2cccc(NS(C)(=O)=O)c2)Nc2c(Cl)cccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.38
CREBBP Q92793 1/20 0.38
OPRM1 P35372 2/20 0.37
KDM1A O60341 2/20 0.37
F11 P03951 1/20 0.36
F7 P08709 1/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP2 O95551 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239526 0.89 GAA (0.42) BRD4KDM1AALDH1A1SMN1; SMN2LMNA
SCHEMBL16239494 0.88 BRD4 (0.39) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL16240072 0.87 CA12 (0.42) BRD4ALDH1A1SMN1; SMN2LMNAGAA
SCHEMBL16239627 0.86 KMT2A (0.41) ALDH1A1LMNAPOLB
SCHEMBL16240075 0.86 L3MBTL1 (0.45) BRD4ALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL16239646 0.85 BRD4 (0.40) BRD4ALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL16239667 0.84 KIF11 (0.40) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL16239481 0.84 BRD4 (0.36) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL2135784 0.81 F11 (0.42) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL16239732 0.80 KDM4E (0.36) ALDH1A1SMN1; SMN2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed