SCHEMBL1625348

SCHEMBL1625348

CCOC(=O)C(C)c1ccc(N)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.55
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
MAOA P21397 1/20 0.55
HTT P42858 2/20 0.51
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
PPID Q08752 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
PPIB P23284 1/20 0.42
PPIA P62937 1/20 0.42
PPIG Q13427 1/20 0.42
TSHR P16473 2/20 0.41
PDE4D Q08499 2/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PRKCZ Q05513 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11037833 0.98 LMNA (0.53) LMNACYP1A2CYP3A4MAOAHTT
SCHEMBL25534680 0.85 ADRB2 (0.41) LMNAHTTSMN1; SMN2TSHRMEN1
SCHEMBL3279844 0.85 KMT2A (0.47) LMNAHTTALDH1A1SMN1; SMN2TSHR
SCHEMBL22838092 0.84 LMNA (0.53) LMNACYP1A2CYP3A4MAOAHTT
SCHEMBL9235662 0.83 ESR1 (0.53) LMNACYP1A2CYP3A4ALDH1A1KDM4E
SCHEMBL9232941 0.83 ESR1 (0.53) LMNACYP1A2CYP3A4ALDH1A1KDM4E
SCHEMBL1792502 0.83 ESR1 (0.53) LMNACYP1A2CYP3A4ALDH1A1KDM4E
SCHEMBL1041487 0.83 LMNA (0.56) LMNACYP1A2CYP3A4MAOAHTT
SCHEMBL11358690 0.83 PTGS2 (0.46) LMNACYP1A2ALDH1A1KDM4ETSHR
SCHEMBL13884372 0.82 EPHX1 (0.45) LMNATSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135831-A Preparation method of alminoprofen intermediate 深圳市华先医药科技有限公司 2021-07-20 CN disclosed
CN-113135831-A Preparation method of alminoprofen intermediate 深圳市华先医药科技有限公司 2021-07-20 CN disclosed
WO-2021027721-A1 IMMUNOMODULATOR 成都先导药物开发股份有限公司 2021-02-18 WO disclosed
CN-111646911-A Method for synthesizing o-aminoacetophenone 广东莱佛士制药技术有限公司 2020-09-11 CN disclosed
US-10752624-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2020-08-25 US disclosed
US-20180305356-A1 NOVEL KINASE INHIBITORS ORIGENIS GMBH (DE) 2018-10-25 US disclosed
US-10000482-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2018-06-19 US disclosed
US-9637491-B2 Pyrazolo[4,3-D]pyrimidines as kinase inhibitors ORIGENIS GMBH (DE) 2017-05-02 US disclosed
US-20150266882-A1 PYRAZOLO[4,3-D]PYRIMIDINES AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2015-09-24 US disclosed
US-20150259340-A1 NOVEL KINASE INHIBITORS ORIGENIS GMBH (DE) 2015-09-17 US disclosed
US-4316850-A ANTINFLAMMATORY AGENTS CIBA-GEIGY CORPORATION (US) 1982-02-23 US disclosed
US-4264619-A Tertiary aminoacids CIBA-GEIGY CORPORATION (US) 1981-04-28 US disclosed
US-4237298-A Aromatic acetic acid derivatives having sulfur atom at alpha-position and process for their preparation SAGAMI CHEMICAL RESEARCH CENTER (JP) 1980-12-02 US disclosed
EP-0011142-A1 Pyrido (2,1-b) quinazolinones, their preparation and pharmaceutical compositions containing them SCHERING AKTIENGESELLSCHAFT (DE) 1980-05-28 EP disclosed
US-4163788-A ANTIINFLAMMATORY CIBA-GEIGY CORPORATION (US) 1979-08-07 US disclosed
US-4144248-A Aromatic acetic acid derivatives having sulfur atom at alpha-position and process for their preparation SAGAMI CHEMICAL RESEARCH CENTER (JP) 1979-03-13 US disclosed
US-4126691-A ANTIINFLAMMATORY CIBA-GEIGY CORPORATION (US) 1978-11-21 US disclosed
US-4118504-A ANALGESICS, ANTIINFLAMMATORY AGENTS Erba, Carlo (IT) 1978-10-03 US disclosed
US-4116972-A ANTI-INFLAMMATORY 1-OXO-ISOINDOLINE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION FUJI CHEMICAL INDUSTRY COMPANY LIMITED (JP) 1978-09-26 US disclosed
US-3997669-A ANTIINFLAMMATORY CIBA-GEIGY CORPORATION (US) 1976-12-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150259340-A1 NOVEL KINASE INHIBITORS LRRK2, MYLK2, MYLK LMNA 3015/4885CYP1A2 3832/4885CYP3A4 4198/4885
US-20150266882-A1 PYRAZOLO[4,3-D]PYRIMIDINES AS KINASE INHIBITORS LRRK2, MYLK2, MYLK LMNA 3243/4885CYP1A2 3276/4885CYP3A4 3280/4885
US-20180305356-A1 NOVEL KINASE INHIBITORS LRRK2, MYLK2, MYLK LMNA 3015/4885CYP1A2 3832/4885CYP3A4 4198/4885
US-10000482-B2 Kinase inhibitors LRRK2, MYLK2, MYLK LMNA 3115/4885CYP1A2 3709/4885CYP3A4 4148/4885
US-10752624-B2 Kinase inhibitors LRRK2, MYLK2, MYLK LMNA 3115/4885CYP1A2 3709/4885CYP3A4 4148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.