SCHEMBL16255461

SCHEMBL16255461

C=CCc1cc(C(c2ccc(OCO)c(CC=C)c2)(C(F)(F)F)C(F)(F)F)ccc1OCO

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
KDM4E B2RXH2 6/20 0.39
LMNA P02545 3/20 0.39
GABRA1 P14867 2/20 0.36
GABRB2 P47870 2/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 5/20 0.35
CNR2 P34972 2/20 0.34
CNR1 P21554 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ELANE P08246 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16255380 0.90 GABRA1 (0.38) PTGDRPTGDR2KDM4ELMNAGABRA1
SCHEMBL195146 0.84 ALDH1A1 (0.43) KDM4ELMNAMAPTALDH1A1MEN1
SCHEMBL194352 0.79 ALDH1A1 (0.38) PTGDRPTGDR2KDM4EGABRA1GABRB2
SCHEMBL16393687 0.79 ELANE (0.35) PTGDRPTGDR2KDM4EGABRA1GABRB2
SCHEMBL21192545 0.79 ALOX5 (0.32) PTGDRPTGDR2GABRA1GABRB2CNR2
SCHEMBL7608902 0.78 ESR1 (0.36) GABRA1GABRB2
SCHEMBL29463283 0.77 GABRA1 (0.56) KDM4ELMNAGABRA1GABRB2MAPT
SCHEMBL29414940 0.77 GABRA1 (0.56) KDM4ELMNAGABRA1GABRB2MAPT
SCHEMBL1055347 0.77 GABRA1 (0.56) KDM4ELMNAGABRA1GABRB2MAPT
SCHEMBL14591648 0.76 PTPN1 (0.34) PTGDRPTGDR2GABRA1GABRB2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889744-B2 Bis-trifluoromethyl honokiol analogs and their use in treating cancers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-11-18 US disclosed