SCHEMBL1627679

SCHEMBL1627679

C=Cc1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]c1=O

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TK2 O00142 5/20 0.74
PYGM P11217 3/20 0.66
SLC28A1 O00337 1/20 0.56
SLC28A2 O43868 1/20 0.56
SLC29A1 Q99808 1/20 0.56
SLC28A3 Q9HAS3 1/20 0.56
P2RY2 P41231 2/20 0.51
DNPH1 O43598 1/20 0.49
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
TK1 P04183 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27786493 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL13597474 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL13447935 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL13413052 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL1532596 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL23083301 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL13252708 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL2587226 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL1532595 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1
SCHEMBL7571099 1.00 TK2 (0.74) TK2PYGMSLC28A1SLC28A2SLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020169140-A1 Combination therapy for reduction of toxicity of chemotherapeutic agents HOLLIS-EDEN PHARMACEUTICALS, INC. 2002-11-14 US claimed
WO-2002069949-A2 COMBINATION THERAPY FOR REDUCTION OF TOXYCITY OF CHEMOTHERAPEUTIC AGENTS PRENDERGAST PATRICK T (IE) 2002-09-12 WO claimed
US-6015573-A TREATMENT OF RESISTANT HERPES VIRUS WITH NUCLEOSIDE PHOSPHATE ESTERS RESOLUTION PERFORMANCE PRODUCTS LLC 2000-01-18 US claimed
US-5879700-A TREATING HERPES VIRUS INFECTIONS HOSTETLER KARL Y (US) 1999-03-09 US claimed
EP-0746319-A4 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER KARL Y (US) 1997-11-05 EP claimed
EP-0746319-A1 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER, Karl Y. (US) 1996-12-11 EP claimed
WO-1994026273-A1 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER KARL Y (US) 1994-11-24 WO claimed
WO-2024124178-A1 METHODS AND APPARATUS FOR TRANSFORM TRAINING AND CODING Beijing Dajia Internet Information Technology Co., Ltd. (CN) 2024-06-13 WO disclosed
US-9549930-B2 Combined systemic and topical treatment of disordered and/or prodromal stage tissue QUADEX PHARMACEUTICALS, LLC (US) 2017-01-24 US disclosed
US-9545408-B2 Combined systemic and topical treatment of disordered tissues QUADEX PHARMACEUTICALS, INC. (US) 2017-01-17 US disclosed
EP-2968228-A1 COMBINED SYSTEMIC AND TOPICAL TREATMENT OF DISORDERED TISSUES Quadex Pharmaceuticals, LLC (US) 2016-01-20 EP disclosed
US-20150374704-A1 COMBINED SYSTEMIC AND TOPICAL TREATMENT OF DISORDERED AND/OR PRODROMAL STAGE TISSUE QUADEX PHARMACEUTICALS, LLC 2015-12-31 US disclosed
CN-105188693-A Combined systemic and topical treatment of disordered tissues QUADEX PHARMACEUTICALS LLC 2015-12-23 CN disclosed
EP-0746319-A4 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER KARL Y (US) 1997-11-05 EP disclosed
EP-0746319-A1 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER, Karl Y. (US) 1996-12-11 EP disclosed
US-5580571-A ACYCLOIR MONO OR DIPHOSPHATE; TOPICAL USE IN HERPES VIRUSINFECTIONS HOSTETLER KARL Y (US) 1996-12-03 US disclosed
WO-1994026273-A1 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER KARL Y (US) 1994-11-24 WO disclosed
WO-1990008128-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS BUNDGAARD HANS (DK) 1990-07-26 WO disclosed
US-4542210-A VIRICIDES, HERPES YAMASA SHOYU KABUSHIKI KAISHA (JP) 1985-09-17 US disclosed
EP-0074101-A1 1-Beta-D-arabinofuranosyl-(E)-5-(2-halogenovinyl) uracil-5'-phosphate, preparation thereof and use thereof Yamasa Shoyu Kabushiki Kaisha (JP) 1983-03-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150374704-A1 COMBINED SYSTEMIC AND TOPICAL TREATMENT OF DISORDERED AND/OR PRODROMAL STAGE TISSUE SAMHD1, CUTA, TK1 TK2 109/4885PYGM 579/4885SLC28A1 24/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.