SCHEMBL16296407

SCHEMBL16296407

O=C1NNN(c2ccc(F)cc2F)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA13 Q8N1Q1 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
OPRM1 P35372 1/20 0.33
AKR1B1 P15121 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
PTGS1 P23219 2/20 0.32
PTGS2 P35354 2/20 0.32
PARK7 Q99497 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16296191 0.72 ALDH1A1 (0.47) L3MBTL1ALDH1A1
SCHEMBL16296173 0.69 DAO (0.33) CA12CA1CA2CA4CA7
SCHEMBL29485045 0.64 MGLL (0.59) GLAL3MBTL1PARK7ALDH1A1
SCHEMBL31662966 0.63 CA12 (0.47) GLACA12CA1CA2CA4
SCHEMBL25291324 0.62 AR (0.48) GLAL3MBTL1OPRM1AKR1B1PTGS1
SCHEMBL8536677 0.62 L3MBTL1 (0.37) GLAL3MBTL1CA12CA1CA2
SCHEMBL8541895 0.62 AR (0.48) CA12CA1CA2CA4CA6
SCHEMBL8723259 0.62 TDP1 (0.42) GLAL3MBTL1CA12CA1CA2
SCHEMBL10362487 0.62 ESR1 (0.45) GLAL3MBTL1CA12CA1CA2
SCHEMBL9779945 0.61 L3MBTL1 (0.36) GLAL3MBTL1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3008055-A1 NOVEL TETRAZOLONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-04-20 EP disclosed
WO-2014198592-A1 NOVEL TETRAZOLONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2014-12-18 WO disclosed