SCHEMBL16486759

SCHEMBL16486759

C[C@@H](C=O)N(C(=O)OC(C)(C)C)c1ncco1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.37
FAAH O00519 1/20 0.31
FFAR2 O15552 1/20 0.31
SSTR4 P31391 1/20 0.31
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16486761 1.00 USP30 (0.37) USP30FAAHFFAR2SSTR4AAK1
SCHEMBL4154644 0.76 PAX8 (0.35) USP30FAAHSSTR4AAK1
SCHEMBL28337730 0.75 FAAH (0.34) USP30FAAHSSTR4AAK1
SCHEMBL7340517 0.74 USP30 (0.37) USP30
SCHEMBL8539792 0.71 SMN1; SMN2 (0.40)
SCHEMBL29245714 0.70 TRPM8 (0.37) FAAHSSTR4
SCHEMBL30366914 0.69 TRPM8 (0.36) FAAHSSTR4
SCHEMBL3989548 0.69 KMT2A (0.40)
SCHEMBL6295154 0.69 SLC6A3 (0.34) USP30
SCHEMBL2791434 0.69 SMN1; SMN2 (0.39) USP30AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145944-A2 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS RQX Pharmaceuticals, Inc. (US) 2017-03-29 EP disclosed
EP-3033352-A1 LINEAR PEPTIDE ANTIBIOTICS RQX Pharmaceuticals, Inc. (US) 2016-06-22 EP disclosed
WO-2015179441-A2 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS RQX PHARMACEUTICALS, INC. (US) 2015-11-26 WO disclosed
WO-2015023898-A1 LINEAR PEPTIDE ANTIBIOTCS RQX PHARMACEUTICALS, INC. (US) 2015-02-19 WO disclosed