SCHEMBL16488279

SCHEMBL16488279

C=Nc1cc(C(F)(F)F)ccc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.46
PDE2A O00408 2/20 0.39
PTPN5 P54829 1/20 0.35
METAP2 P50579 1/20 0.35
LRRK2 Q5S007 1/20 0.34
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.32
XBP1 P17861 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
KIF11 P52732 4/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 2/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22620411 0.78 PDE2A (0.41) PDE2APTPN5MAPTKIF11ALDH1A1
SCHEMBL31135808 0.75 CES2 (0.46) CES2PDE2APTPN5METAP2CYP3A4
SCHEMBL7057873 0.75 CES2 (0.42) CES2PDE2APTPN5METAP2TSHR
SCHEMBL12535901 0.75 CES2 (0.46) CES2PDE2APTPN5METAP2CYP3A4
SCHEMBL28770910 0.75 PDE2A (0.50) CES2PDE2APTPN5METAP2TSHR
SCHEMBL22620302 0.73 ADRA2A (0.40) PDE2APTPN5NPSR1KIF11ALDH1A1
SCHEMBL20052480 0.73 L3MBTL1 (0.44) LRRK2MAPK1MAPTNPSR1CYP3A4
SCHEMBL6061078 0.72 CES2 (0.56) CES2PDE2APTPN5TSHRMAPK1
SCHEMBL18979040 0.72 CES2 (0.40) CES2PDE2AMETAP2LRRK2MAPT
SCHEMBL31571863 0.72 ALDH1A1 (0.41) CES2TSHRMAPK1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238152-B1 PROCESSES FOR PREPARATION OF DUTASTERIDE GADOR SA (AR) 2015-02-18 EP disclosed