SCHEMBL16600237

SCHEMBL16600237

COC(=O)c1ccc(N2CCN(c3ccc(Cl)c(Cl)c3)CC2)cc1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 13/20 0.61
SMN1; SMN2 Q16637 7/20 0.61
RAB9A P51151 1/20 0.56
HTT P42858 4/20 0.52
MAPK1 P28482 1/20 0.52
TP53 P04637 3/20 0.51
POLB P06746 1/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 4/20 0.47
LMNA P02545 3/20 0.47
TSHR P16473 1/20 0.47
PANK3 Q9H999 1/20 0.46
KDM4E B2RXH2 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALOX12 P18054 1/20 0.46
RECQL P46063 2/20 0.45
SIRT6 Q8N6T7 1/20 0.45
THRB P10828 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16600119 0.92 ALDH1A1 (0.52) MAPTSMN1; SMN2RAB9AHTTMEN1
SCHEMBL16599909 0.88 SIRT6 (0.46) MAPTSMN1; SMN2RAB9AHTTTP53
SCHEMBL16600104 0.88 CYP1A2 (0.52) MAPTSMN1; SMN2RAB9AHTTMAPK1
SCHEMBL16609018 0.86 SIRT6 (0.47) MAPTSMN1; SMN2RAB9AHTTMEN1
SCHEMBL16599996 0.86 KMT2A (0.48) MAPTSMN1; SMN2TP53KMT2AALDH1A1
SCHEMBL16600133 0.85 WDR5 (0.47) MAPTSMN1; SMN2RAB9AMEN1KMT2A
SCHEMBL1890774 0.85 SIRT6 (0.61) MAPTSMN1; SMN2RAB9AHTTMAPK1
SCHEMBL20976884 0.85 MAPT (0.51) MAPTSMN1; SMN2RAB9AMAPK1TP53
SCHEMBL16608992 0.83 RAB9A (0.53) MAPTSMN1; SMN2RAB9ATP53MEN1
SCHEMBL16600000 0.83 DRD2 (0.47) KMT2AALDH1A1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015048306-A1 NOVEL AGENTS TARGETING CYP51 THE SCRIPPS RESEARCH INSTITUTE (US) 2015-04-02 WO disclosed