SCHEMBL1660370

SCHEMBL1660370

C=Cc1cc(-c2ccc([C]=O)o2)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
SLC6A1 P30531 1/20 0.31
SLC9A1 P19634 1/20 0.31
RXRA P19793 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12521317 0.77 NR4A1 (0.45) KDM4EALDH1A1SLC9A1RXRACYP1A2
SCHEMBL2323764 0.76 KDM4E (0.52) KDM4EALDH1A1SLC9A1RXRACYP1A2
SCHEMBL1661873 0.75 NOTUM (0.46) KDM4EALDH1A1SLC6A1
SCHEMBL2318440 0.75 CYP1A1 (0.42) CYP1A2CYP2C19
SCHEMBL347778 0.68 CES2 (0.41) ALDH1A1
SCHEMBL6009742 0.65 MEN1 (0.45) KDM4E
SCHEMBL7325347 0.65 AR (0.35) KDM4EALDH1A1SLC9A1RXRACYP1A2
SCHEMBL1063612 0.64 KDM4E (0.54) KDM4EALDH1A1SLC6A1RXRACYP2C19
SCHEMBL12328697 0.64 KDM4E (0.63) KDM4EALDH1A1SLC9A1RXRACYP1A2
SCHEMBL21012216 0.64 KIF11 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed
WO-2010002209-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2010-01-07 WO disclosed