SCHEMBL16610416

SCHEMBL16610416

CCCCOc1cc(/C=C/C(=O)NC)cc(C(F)(F)F)c1OCCCC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43
CYP1A2 P05177 3/20 0.43
CYP2C19 P33261 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
APP P05067 2/20 0.40
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
CNR2 P34972 3/20 0.38
PSMB11 A5LHX3 1/20 0.37
PSMA7 O14818 1/20 0.37
PSMB1 P20618 1/20 0.37
PSMA1 P25786 1/20 0.37
PSMA2 P25787 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610417 0.87 KDM4E (0.48) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL16610426 0.84 THRA (0.40) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL16610411 0.83 APP (0.41) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL16610407 0.79 ALDH1A1 (0.39) KDM4EALDH1A1POLBMEN1MAPT
SCHEMBL16610335 0.75 TRPV1 (0.47) HTR1AHTR2CHTR2ASLC6A4HTR7
SCHEMBL16610334 0.75 THRB (0.44) HTR1AHTR2CKDM4EALDH1A1CYP3A4
SCHEMBL28818999 0.70 PELI1 (0.46) CYP1A2CYP2C19KDM4EALDH1A1CYP3A4
SCHEMBL16610343 0.70 PELI1 (0.46) CYP1A2CYP2C19KDM4EALDH1A1CYP3A4
SCHEMBL9112337 0.70 ABCG2 (0.56) KDM4EALDH1A1MAPTACHE
SCHEMBL21133746 0.69 CYP1A2 (0.42) HTR1AHTR2CHTR2ASLC6A4HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed