SCHEMBL16610426

SCHEMBL16610426

CCCCOc1cc(/C=C/C(=O)N(C)C)cc(C(F)(F)F)c1OCCCC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 2/20 0.40
THRB P10828 2/20 0.40
APP P05067 4/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HTR1A P08908 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALOX5 P09917 3/20 0.36
AKR1C3 P42330 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610411 0.90 APP (0.41) THRATHRBAPPMEN1KMT2A
SCHEMBL16610417 0.87 KDM4E (0.48) THRATHRBAPPMEN1KMT2A
SCHEMBL16610416 0.84 HTR1A (0.43) APPMEN1KMT2AHTR1AHTR2C
SCHEMBL16610407 0.79 ALDH1A1 (0.39) THRATHRBMEN1KMT2AKDM4E
SCHEMBL16610334 0.75 THRB (0.44) THRATHRBAPPMEN1KMT2A
SCHEMBL16610382 0.70 GABBR2 (0.40) APPCYP1A2CYP3A4ALOX5PTGES
SCHEMBL9112337 0.70 ABCG2 (0.56) KDM4EALDH1A1CYP1A1CYP1B1SMN1; SMN2
SCHEMBL21133746 0.69 CYP1A2 (0.42) APPHTR1AHTR2CHTR2ASLC6A4
SCHEMBL16610335 0.69 TRPV1 (0.47) THRBAPPHTR1AHTR2CHTR2A
SCHEMBL16610333 0.68 APP (0.36) THRATHRBAPPKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed