SCHEMBL16612728

SCHEMBL16612728

NC(=O)c1[c]cn(CCc2cccc(F)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.43
SLC6A3 Q01959 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
HTR2A P28223 1/20 0.40
MAOB P27338 1/20 0.40
PARP10 Q53GL7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
DAO P14920 1/20 0.39
SLC1A1 P43005 2/20 0.39
ATM Q13315 1/20 0.38
PARP1 P09874 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520701 0.87 L3MBTL1 (0.50) NR3C2MAOBPARP10L3MBTL1SLC1A1
SCHEMBL14699373 0.84 ADORA2A (0.47) L3MBTL1PARP1
SCHEMBL16612943 0.82 SIGMAR1 (0.47) NR3C2TAAR1MAOBDAOPARP1
SCHEMBL16612828 0.80 SIRT2 (0.39) MAOBPARP10PARP1
SCHEMBL15520668 0.76 HDAC1 (0.34) L3MBTL1PARP1
SCHEMBL16612788 0.74 MPO (0.56) HTR2A
SCHEMBL15520768 0.73 LMNA (0.40) MAOBPARP10MAPT
SCHEMBL14699416 0.73 HTT (0.43) L3MBTL1
SCHEMBL1718132 0.73 PARP1 (0.48) L3MBTL1PARP1
SCHEMBL14699254 0.72 HDAC1 (0.44) PARP10PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed